Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50024909
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50117090((E,E)-Psammaplin A | 3-(3-Bromo-4-hydroxy-phenyl)-...)
Affinity DataEC50:  5.70E+3nMAssay Description:Activation of PPARgamma (unknown origin) transfected in human MCF7 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataEC50:  5.00E+4nMAssay Description:Activation of GAL4 fused human PPARgamma ligand binding domain transfected in african green monkey CV1 cells by CAT reporter assayMore data for this Ligand-Target Pair