Affinity DataKi: 244nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 319nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 670nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.42E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.78E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by ChEMBL
Asahi Kasei Pharma
Curated by ChEMBL
Affinity DataEC50: 1.80nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 16.4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by ChEMBL
Asahi Kasei Pharma
Curated by ChEMBL
Affinity DataEC50: 3.30E+3nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by ChEMBL
Asahi Kasei Pharma
Curated by ChEMBL
Affinity DataEC50: 135nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by ChEMBL
Asahi Kasei Pharma
Curated by ChEMBL
Affinity DataEC50: 77.4nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 15.4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.11E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.58E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by ChEMBL
Asahi Kasei Pharma
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 72.9nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.12E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by ChEMBL
Asahi Kasei Pharma
Curated by ChEMBL
Affinity DataEC50: 67nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.01E+4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by ChEMBL
Asahi Kasei Pharma
Curated by ChEMBL
Affinity DataEC50: 5.10E+3nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 9.59E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by ChEMBL
Asahi Kasei Pharma
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair