Compile Data Set for Download or QSAR
maximum 50k data
Found 37 Enz. Inhib. hit(s) with all data for entry = 50017792
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186560(1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimi...)
Affinity DataIC50:  3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186557(1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimi...)
Affinity DataIC50:  3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186566(3-(5-((5-tert-butylisoxazol-3-yl)carbamoyl)-2-meth...)
Affinity DataIC50:  4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186535(3-(5-hydroxy-2-methylphenyl)-1-methyl-1-(6-(4-morp...)
Affinity DataIC50:  4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186556(3-(2,6-dichlorophenyl)-1-methyl-1-(6-(4-(4-methylp...)
Affinity DataIC50:  6nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186554(3-(2-chloro-6-methylphenyl)-1-methyl-1-(6-(4-(4-me...)
Affinity DataIC50:  9nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186537(3-(2-chloro-6-methylphenyl)-1-(6-(4-(2-(diethylami...)
Affinity DataIC50:  28nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186558(1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimi...)
Affinity DataIC50:  32nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186541(3-(5-(benzo[b]thiophene-2-carboxamido)-2-methylphe...)
Affinity DataIC50:  52nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186538(3-(2,6-dichlorophenyl)-1-(6-(4-(2-(diethylamino)et...)
Affinity DataIC50:  87nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186567(3-(2-chloro-6-(trifluoromethyl)phenyl)-1-(6-(4-(2-...)
Affinity DataIC50:  96nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186546(1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimi...)
Affinity DataIC50:  149nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186569(3-(2,6-dichlorophenyl)-1-(3-(dimethylamino)propyl)...)
Affinity DataIC50:  155nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186548(3-(2-chloro-6-methylphenyl)-1-methyl-1-(6-(4-morph...)
Affinity DataIC50:  190nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186543(3-(2,6-dichlorophenyl)-1-(6-(4-(2-(diethylamino)et...)
Affinity DataIC50:  229nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186540(3-(2,6-dichlorophenyl)-1-(4-methylpiperazin-1-yl)-...)
Affinity DataIC50:  230nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186539(3-(2,6-dichlorophenyl)-1-methyl-1-(6-(4-morpholino...)
Affinity DataIC50:  301nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186565(1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimi...)
Affinity DataIC50:  418nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186542(3-(2-chlorophenyl)-1-methyl-1-(6-(4-(4-methylpiper...)
Affinity DataIC50:  708nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186553(3-(2-chloro-6-methylphenyl)-1-(6-(4-(diethylamino)...)
Affinity DataIC50:  971nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186568(1-benzyl-3-(2-chloro-6-methylphenyl)-1-(6-(4-fluor...)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186545(3-(2-chlorophenyl)-1-(6-(4-fluorophenylamino)pyrim...)
Affinity DataIC50:  1.82E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186534(3-(2,6-dichlorophenyl)-1-(3-(dimethylamino)propyl)...)
Affinity DataIC50:  2.35E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186561(1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimi...)
Affinity DataIC50:  2.58E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186555(3-(2-chlorophenyl)-1-(6-(4-(diethylamino)phenylami...)
Affinity DataIC50:  3.13E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186549(3-(2,6-dichlorophenyl)-1-(6-(4-fluorophenylamino)p...)
Affinity DataIC50:  3.86E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186551(3-(2-chlorophenyl)-1-methyl-1-(6-(4-morpholinophen...)
Affinity DataIC50:  4.29E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186564(3-(2-chlorophenyl)-1-(6-(4-(diethylamino)phenylami...)
Affinity DataIC50:  4.49E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186570(3-(2,6-dichlorophenyl)-1-(6-(3-(dimethylamino)prop...)
Affinity DataIC50:  5.99E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186547(3-(2,6-dichlorophenyl)-1-(4-(2-(diethylamino)ethox...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186563(1-(4-(dimethylamino)benzyl)-3-(2-chlorophenyl)-1-(...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186550(3-(2,6-dichlorophenyl)-1-methyl-1-(6-(2-morpholino...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186552(3-(2,6-dichlorophenyl)-1-(6-(4-morpholinophenylami...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186562(3-(2,6-dichlorophenyl)-1-methyl-1-(6-(tetrahydro-2...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186544(1-(6-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186559(1-benzyl-3-(2-chlorophenyl)-1-(6-(4-(diethylamino)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50186536(3-(2,6-dichlorophenyl)-1-(6-(2-(diethylamino)ethyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed