Compile Data Set for Download or QSAR
maximum 50k data
Found 94 Enz. Inhib. hit(s) with all data for entry = 50017843
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  38nMAssay Description:Inhibition of DPP4 in Sprague-Dawley rat plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187283((2R,5S)-1-(2-(1-(ethoxymethyl)cyclopentylamino)ace...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187258((2S,5R)-1-[2-(hexahydro-2,5-methano-pentalen-3a-yl...)
Affinity DataIC50:  72nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187263((2S,5R)-1-[2-(3-hydroxy-adamantan-1-ylamino)-acety...)
Affinity DataIC50:  74nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187275((2R,5S)-1-(2-(1-(methoxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  84nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187261((2R,5S)-1-(2-(1-(butoxymethyl)cyclopentylamino)ace...)
Affinity DataIC50:  91nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  92nMAssay Description:Inhibition of DPP4 in cynomolgus monkey plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  104nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187268((2S,5R)-1-[2-(adamantan-1-ylamino)-acetyl]-pyrroli...)
Affinity DataIC50:  106nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  109nMAssay Description:Inhibition of DPP4 in beagle dog plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  109nMAssay Description:Inhibition of DPP4 in beagle dog plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187294((2R,5S)-1-(2-(1-(propoxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  123nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187305((2R,5S)-1-(2-(1-phenylcyclobutylamino)acetyl)pyrro...)
Affinity DataIC50:  164nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187271((2R,5S)-1-(2-(1-methylcyclopentylamino)acetyl)pyrr...)
Affinity DataIC50:  201nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187265((2R,5S)-1-(2-(2,4,4-trimethylpentan-2-ylamino)acet...)
Affinity DataIC50:  208nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187274(CHEMBL211024 | exo-(2R,5S)-1-(2-(bicyclo[2.2.1]hep...)
Affinity DataIC50:  237nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187276((2R,5S)-1-(2-(2-phenylpropan-2-ylamino)acetyl)pyrr...)
Affinity DataIC50:  261nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187269((2R,5S)-1-(2-(1-(isobutoxymethyl)cyclopentylamino)...)
Affinity DataIC50:  454nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187260((2R,5S)-1-(2-(1-(4-fluorophenyl)-2-methylpropan-2-...)
Affinity DataIC50:  651nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187279((2R,5S)-1-(2-(tert-butylamino)acetyl)pyrrolidine-2...)
Affinity DataIC50:  663nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187273((2R,5S)-1-(2-(1-(hydroxymethyl)cyclohexylamino)ace...)
Affinity DataIC50:  687nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187280((2R,5S)-1-(2-(1-methylcyclohexylamino)acetyl)pyrro...)
Affinity DataIC50:  689nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187298((2R,5S)-1-(2-(1-(cyclohexyloxymethyl)cyclopentylam...)
Affinity DataIC50:  702nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187303((2R,5S)-1-(2-(1,3-dimethylcyclopentylamino)acetyl)...)
Affinity DataIC50:  771nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187289((2R,5S)-1-(2-(2-(hydroxymethyl)-2,3-dihydro-1H-ind...)
Affinity DataIC50:  875nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187302((2R,5S)-1-(2-(1-(2-methoxyethyl)cyclopentylamino)a...)
Affinity DataIC50:  955nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187278((2R,5S)-1-(2-(1-hydroxy-2-methylpropan-2-ylamino)a...)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187301((2R,5S)-1-(2-(1-benzylcyclobutylamino)acetyl)pyrro...)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187293((2R,5S)-1-(2-(4-(hydroxymethyl)-tetrahydro-2H-pyra...)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187290((2R,5S)-1-(2-(1-(3,3-dimethyl-2-oxobutyl)cyclopent...)
Affinity DataIC50:  1.86E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187259((2R,5S)-1-(2-(1,2,2-trimethylcyclopentylamino)acet...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187262(CHEMBL209933 | methyl 1-(2-((2R,5S)-2,5-dicyanopyr...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187264((2R,5S)-1-(2-(2,3,3-trimethylbutan-2-ylamino)acety...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187272((2R,5S)-1-(2-(2,3-dimethylbutan-2-ylamino)acetyl)p...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187277((2S,5R)-1-[2-(3,5,7-trifluoro-adamantan-1-ylamino)...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187281((2R,5S)-1-(2-(1-ethynylcyclohexylamino)acetyl)pyrr...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187282((2R,5S)-1-(2-(1-(2-hydroxyethyl)cyclopentylamino)a...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187285((2R,5S)-1-(2-(1-(3-hydroxypropyl)cyclohexylamino)a...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187286((2R,5S)-1-(2-(3-methyl-tetrahydrothiophen-3-ylamin...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187288(1-(2-((2R,5S)-2,5-dicyanopyrrolidin-1-yl)-2-oxoeth...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187287((2R,5S)-1-(2-(1-benzylcyclohexylamino)acetyl)pyrro...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187291((2R,5S)-1-(2-(tert-pentylamino)acetyl)pyrrolidine-...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187292((2R,5S)-1-(2-(2,2,5-trimethyl-1,3-dioxan-5-ylamino...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187295((2R,5S)-1-(2-(3-methylpentan-3-ylamino)acetyl)pyrr...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187296((2R,5S)-1-(2-(1-methyl-3-tert-pentylcyclopentylami...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187300((2R,5S)-1-(2-(1-ethylcyclohexylamino)acetyl)pyrrol...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187304((2R,5S)-1-(2-((3S,4R)-1,3,4-trimethylcyclopentylam...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187263((2S,5R)-1-[2-(3-hydroxy-adamantan-1-ylamino)-acety...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187261((2R,5S)-1-(2-(1-(butoxymethyl)cyclopentylamino)ace...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187268((2S,5R)-1-[2-(adamantan-1-ylamino)-acetyl]-pyrroli...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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