Compile Data Set for Download or QSAR
maximum 50k data
Found 35 Enz. Inhib. hit(s) with all data for entry = 50037701
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50422861(CHEMBL2304221)
Affinity DataEC50:  0.800nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50069108(1-{[(2R)-1-{2,3-dihydrospiro[indene-1,4'-piperidin...)
Affinity DataEC50:  14nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187307(1-{[(2R)-3-(benzyloxy)-1-oxo-1-{2H-spiro[1-benzoth...)
Affinity DataEC50:  10nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370712(CHEMBL1793862)
Affinity DataEC50:  3nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187310(1-((R)-1-((S)-3a-benzyl-2-ethyl-3-oxo-2,3,3a,4,6,7...)
Affinity DataEC50:  4nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187308(1-{[(2R)-3-(benzyloxy)-1-{2,3-dihydrospiro[indene-...)
Affinity DataEC50:  17nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187312(1-methyl-1-{[(2R)-1-oxo-5-phenyl-1-{2H-spiro[1-ben...)
Affinity DataEC50:  4.80nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187313(1-methyl-1-((R)-1-{2'-[(3-methyl-ureido)-methyl]-b...)
Affinity DataEC50:  1nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187314(1-methyl-1-{[(2R)-1-oxo-5-phenyl-1-{2H-spiro[1-ben...)
Affinity DataEC50:  2.70nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187315(1-{[(2R)-1-{1,1-dioxo-2H-spiro[1-benzothiophene-3,...)
Affinity DataEC50:  6nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187317(1-{[(2R)-1-{2,3-dihydrospiro[indene-1,4'-piperidin...)
Affinity DataEC50:  22nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187318(1-((R)-1-((S)-3a-benzyl-2-methyl-3-oxo-2,3,3a,4,6,...)
Affinity DataEC50:  3nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187316(1-{[(2R)-1-[(3R)-3-hydroxy-2,3-dihydrospiro[indene...)
Affinity DataEC50:  0.600nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187319(1-{[(2R)-1-{1,1-dioxo-2H-spiro[1-benzothiophene-3,...)
Affinity DataEC50:  1.10nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187320(1-{[(2R)-3-(benzyloxy)-1-oxo-1-{2H-spiro[1-benzofu...)
Affinity DataEC50:  8.5nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187322(1-{[(2R)-1-{2,3-dihydrospiro[indene-1,4'-piperidin...)
Affinity DataEC50:  10nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187321(1-((R)-1-((S)-3a-benzyl-3-oxo-2,3,3a,4,6,7-hexahyd...)
Affinity DataEC50:  3nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187323((R,E)-6-((1-((2-(methylsulfonamido)phenethyl)(meth...)
Affinity DataEC50:  18nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50066816((E)-2-methyl-6-(methyl((R)-1-(methyl((R)-1-(methyl...)
Affinity DataEC50:  3nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187325(1-((R)-1-{2'-[(3-ethyl-ureido)-methyl]-biphenyl-4-...)
Affinity DataEC50:  6nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370713(CHEMBL1162926)
Affinity DataEC50:  3nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187326((R)-5-amino-N,5-dimethyl-N-(1-(methyl(2-(thiophen-...)
Affinity DataEC50:  7.5nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50065107((R)-1-[(R)-2-(2-amino-2-methyl-propionylamino)-3-(...)
Affinity DataEC50:  1.60nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187327(1-{[(2R)-1-{1,1-dioxo-2H-spiro[1-benzothiophene-3,...)
Affinity DataEC50:  2.10nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370714(CHEMBL1161827)
Affinity DataEC50:  2nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187329((R,E)-6-((1-((2-(2-hydroxyethoxy)phenethyl)(methyl...)
Affinity DataEC50:  5nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187330((R)-N,5-dimethyl-N-(1-(methyl(2-(thiophen-2-yl)eth...)
Affinity DataEC50:  0.800nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187332(1-{[(2R)-3-(1H-indol-3-yl)-1-oxo-1-{2H-spiro[1-ben...)
Affinity DataEC50:  5.60nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187331((R,E)-6-((1-((2-(2-hydroxyethoxy)phenethyl)(methyl...)
Affinity DataEC50:  5nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370715(CHEMBL1161826)
Affinity DataEC50:  8.5nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187333((E)-4-({(R)-2-biphenyl-4-yl-1-[methyl-(2-thiophen-...)
Affinity DataEC50:  5nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187335(1-methyl-1-{[(2R)-1-oxo-4-phenyl-1-{2H-spiro[1-ben...)
Affinity DataEC50:  57nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187336(2-amino-N-[(2R)-3-(benzyloxy)-1-[(3R)-3-hydroxy-2,...)
Affinity DataEC50:  1.30nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187337(1-((R)-1-{2'-[3-(2-hydroxy-ethyl)-ureidomethyl]-bi...)
Affinity DataEC50:  2nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50187306(1-{[(2R)-3-(benzyloxy)-1-{1,1-dioxo-2H-spiro[1-ben...)
Affinity DataEC50:  5nMAssay Description:Activity at human GHS-R1a receptor in rat pitutary cells assessed as GH releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed