Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50017862
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187669(CHEMBL207208 | N-(4-methoxy-phenyl)-2-cyclopentyl-...)
Affinity DataKi:  410nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50011596((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
Affinity DataKi:  786nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187670(CHEMBL210380 | N-(4-methyl-phenyl)-2-cyclopentyl-1...)
Affinity DataKi:  1.19E+3nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187671(CHEMBL378047 | N-(4-chloro-phenyl)-2-cyclopentyl-1...)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50011596((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
Affinity DataKi:  3.15E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50011596((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
Affinity DataKi:  3.42E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187670(CHEMBL210380 | N-(4-methyl-phenyl)-2-cyclopentyl-1...)
Affinity DataKi:  3.85E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187669(CHEMBL207208 | N-(4-methoxy-phenyl)-2-cyclopentyl-...)
Affinity DataKi:  4.17E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187672(CHEMBL207209 | N-(3,4-dichloro-phenyl)-2-cyclopent...)
Affinity DataKi:  4.69E+3nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187670(CHEMBL210380 | N-(4-methyl-phenyl)-2-cyclopentyl-1...)
Affinity DataKi:  5.22E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187672(CHEMBL207209 | N-(3,4-dichloro-phenyl)-2-cyclopent...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187671(CHEMBL378047 | N-(4-chloro-phenyl)-2-cyclopentyl-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187672(CHEMBL207209 | N-(3,4-dichloro-phenyl)-2-cyclopent...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187671(CHEMBL378047 | N-(4-chloro-phenyl)-2-cyclopentyl-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187669(CHEMBL207208 | N-(4-methoxy-phenyl)-2-cyclopentyl-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed