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Found 70 Enz. Inhib. hit(s) with all data for entry = 50017920
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188394((+)-N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]propyl)...)
Affinity DataKi:  0.270nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.350nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.390nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188394((+)-N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]propyl)...)
Affinity DataKi:  0.410nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188417(CHEMBL377101 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  0.470nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188394((+)-N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]propyl)...)
Affinity DataKi:  0.5nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188406(CHEMBL207745 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  0.740nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188408(CHEMBL207625 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  0.860nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188402(CHEMBL379616 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  1.02nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188423(CHEMBL206472 | beta,beta-dimethylmelatonin)
Affinity DataKi:  1.12nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188411(CHEMBL426127 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  1.15nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188394((+)-N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]propyl)...)
Affinity DataKi:  1.22nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188420(CHEMBL208307 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  1.29nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188412(CHEMBL210147 | beta-methylmelatonin)
Affinity DataKi:  1.67nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188423(CHEMBL206472 | beta,beta-dimethylmelatonin)
Affinity DataKi:  2.75nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188412(CHEMBL210147 | beta-methylmelatonin)
Affinity DataKi:  2.94nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188400(CHEMBL207960 | N-(2-[5-methoxy-1H-indol-3-yl]-2,2-...)
Affinity DataKi:  3.30nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188417(CHEMBL377101 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  4.27nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188401(CHEMBL424693 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  4.40nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188402(CHEMBL379616 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  4.90nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188394((+)-N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]propyl)...)
Affinity DataKi:  5.48nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188411(CHEMBL426127 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  6.03nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188422(CHEMBL209712 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  7.5nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188394((+)-N-(2-[5-methoxy-1-methyl-1H-indol-3-yl]propyl)...)
Affinity DataKi:  7.71nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188400(CHEMBL207960 | N-(2-[5-methoxy-1H-indol-3-yl]-2,2-...)
Affinity DataKi:  8.20nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188406(CHEMBL207745 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  8.51nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188408(CHEMBL207625 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  10.6nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188420(CHEMBL208307 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  11.5nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188413(CHEMBL206790 | N-(2-[5-methoxy-1H-indol-3-yl]-2,2-...)
Affinity DataKi:  28.9nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188416(CHEMBL207420 | N-(2-[5-methoxy-1H-indol-3-yl]-2,2-...)
Affinity DataKi:  32nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188403(CHEMBL382439 | N-(2-(5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  33.1nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188401(CHEMBL424693 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  34nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188410(CHEMBL377871 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  39nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188397(CHEMBL207676 | N-(2-[5-methoxy-1H-indol-3-yl]-2,2-...)
Affinity DataKi:  57.4nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188413(CHEMBL206790 | N-(2-[5-methoxy-1H-indol-3-yl]-2,2-...)
Affinity DataKi:  57.8nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188395(CHEMBL377809 | N-(2-[5-methoxy-1H-indol-3-yl]-2,2-...)
Affinity DataKi:  62.2nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188416(CHEMBL207420 | N-(2-[5-methoxy-1H-indol-3-yl]-2,2-...)
Affinity DataKi:  65.7nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188414(CHEMBL379403 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  66.1nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188419(CHEMBL379413 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  72nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188396(CHEMBL206419 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  85.1nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188410(CHEMBL377871 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  86nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188424(CHEMBL209711 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  90nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188404(CHEMBL382555 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  102nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188397(CHEMBL207676 | N-(2-[5-methoxy-1H-indol-3-yl]-2,2-...)
Affinity DataKi:  116nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188405(CHEMBL382579 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  138nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188414(CHEMBL379403 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  148nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188403(CHEMBL382439 | N-(2-(5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  170nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188424(CHEMBL209711 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  176nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188422(CHEMBL209712 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  212nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50188415(CHEMBL206471 | N-(2-[5-methoxy-1-methyl-1H-indol-3...)
Affinity DataKi:  257nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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