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Found 29 Enz. Inhib. hit(s) with all data for entry = 50037738
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  226nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat DAT expressed in D8 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190380(CHEMBL374492 | bip-tyr-thr-pro-thr(obzl)-gly)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  400nMAssay Description:Inhibition of rat SERT-mediated serotonin uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190380(CHEMBL374492 | bip-tyr-thr-pro-thr(obzl)-gly)
Affinity DataIC50:  494nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat DAT expressed in D8 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  900nMAssay Description:Inhibition of rat NET-mediated norepinephrine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190379(CHEMBL439332 | bip-tyr-thr-ala-pro-phe)
Affinity DataIC50:  900nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190385(CHEMBL219358 | bip-tyr-thr-pro-ala-thr(obzl)-gly)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190387(CHEMBL428483 | bip-tyr-thr-pro-lys-thr(obzl)-gly)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190388(CHEMBL385983 | bip-tyr(3bzl)-thr-pro-lys-thr)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190389(CHEMBL277108 | bip-tyr-ala-pro-lys-thr(obzl)-gly)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190382(CHEMBL379496 | bip-tyr-thr-pro-lys-thr)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190375(CHEMBL269579 | bip-tyr-thr(obzl)-pro-lys-thr-gly)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190379(CHEMBL439332 | bip-tyr-thr-ala-pro-phe)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of rat NET-mediated norepinephrine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190379(CHEMBL439332 | bip-tyr-thr-ala-pro-phe)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of rat SERT-mediated serotonin uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190380(CHEMBL374492 | bip-tyr-thr-pro-thr(obzl)-gly)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of rat NET-mediated norepinephrine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190380(CHEMBL374492 | bip-tyr-thr-pro-thr(obzl)-gly)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of rat SERT-mediated serotonin uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190376(CHEMBL383931 | bip-ala-thr-pro-lys-thr(obzl)-gly)
Affinity DataIC50:  1.73E+5nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190383(CHEMBL411570 | nal2-tyr-thr-pro-lys-thr(obzl)-gly)
Affinity DataIC50:  1.84E+5nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190384(CHEMBL218952 | nal1-tyr-thr-pro-lys-thr(obzl)-gly)
Affinity DataIC50:  1.99E+5nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190386(CHEMBL409615 | bpa-tyr-thr-pro-lys-thr(obzl)-gly)
Affinity DataIC50:  2.39E+5nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190379(CHEMBL439332 | bip-tyr-thr-ala-pro-phe)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of mouse GAT1-mediated gamma-aminobutyric acid uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190380(CHEMBL374492 | bip-tyr-thr-pro-thr(obzl)-gly)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of mouse GAT1-mediated gamma-aminobutyric acid uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190382(CHEMBL379496 | bip-tyr-thr-pro-lys-thr)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of rat NET-mediated norepinephrine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190378(CHEMBL219062 | bip-tyr-thr-ala-lys-thr(obzl)-gly)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190377(CHEMBL212513 | phe-phe-tyr-thr-pro-lys-thr)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190382(CHEMBL379496 | bip-tyr-thr-pro-lys-thr)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of rat SERT-mediated serotonin uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190382(CHEMBL379496 | bip-tyr-thr-pro-lys-thr)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of mouse GAT1-mediated gamma-aminobutyric acid uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50190381(CHEMBL209752 | bip-tyr-thr-ala-thr(obzl)-gly)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed