Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50018086
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)
Affinity DataIC50:  0.970nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)
Affinity DataIC50:  0.990nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191053(1-ethyl-3-(3-oxo-3-((1-phenethylpiperidin-4-yl)(ph...)
Affinity DataIC50:  30nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)
Affinity DataIC50:  35nMAssay Description:Activity at delta opioid receptor by MVD assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)
Affinity DataIC50:  42nMAssay Description:Activity at mu opioid receptor by GPI/LMMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191057(CHEMBL214657 | N-(1-phenethylpiperidin-4-yl)-N-phe...)
Affinity DataIC50:  146nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191055(3-(1,3-dioxoisoindolin-2-yl)-N-(1-phenethylpiperid...)
Affinity DataIC50:  217nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191058(CHEMBL214285 | N-(1-phenethyl-piperidin-4-yl)-N-ph...)
Affinity DataIC50:  450nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191058(CHEMBL214285 | N-(1-phenethyl-piperidin-4-yl)-N-ph...)
Affinity DataIC50:  451nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191060(3-acetamido-N-(1-phenethylpiperidin-4-yl)-N-phenyl...)
Affinity DataIC50:  1.03E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191054(3-amino-N-(1-phenethylpiperidin-4-yl)-N-phenylprop...)
Affinity DataIC50:  2.08E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191059(2-acetylamino-N-{2-[(1-phenethyl-piperidin-4-yl)-p...)
Affinity DataIC50:  2.68E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM21114(3-{phenyl[1-(2-phenylethyl)piperidin-4-yl]carbamoy...)
Affinity DataIC50:  5.40E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191053(1-ethyl-3-(3-oxo-3-((1-phenethylpiperidin-4-yl)(ph...)
Affinity DataIC50:  6.65E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191059(2-acetylamino-N-{2-[(1-phenethyl-piperidin-4-yl)-p...)
Affinity DataIC50:  7.60E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191060(3-acetamido-N-(1-phenethylpiperidin-4-yl)-N-phenyl...)
Affinity DataIC50:  8.40E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM21114(3-{phenyl[1-(2-phenylethyl)piperidin-4-yl]carbamoy...)
Affinity DataIC50:  9.40E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191057(CHEMBL214657 | N-(1-phenethylpiperidin-4-yl)-N-phe...)
Affinity DataIC50:  1.21E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50191054(3-amino-N-(1-phenethylpiperidin-4-yl)-N-phenylprop...)
Affinity DataIC50:  1.30E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed