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Found 8 Enz. Inhib. hit(s) with all data for entry = 50018319
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194360((E)-thyl-1-methyl-6,7-dihydro-1H-indol-4(5H)-one O...)
Affinity DataIC50:  21nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194358((E)--2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-phe...)
Affinity DataIC50:  67nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194357((E)--2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-4-f...)
Affinity DataIC50:  275nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194361((E)--2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-4-(...)
Affinity DataIC50:  350nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194362((E)-1-(4-((3-ethyl-1,2-dimethyl-6,7-dihydro-1H-ind...)
Affinity DataIC50:  368nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194359((E)--2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-2-(...)
Affinity DataIC50:  547nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194360((E)-thyl-1-methyl-6,7-dihydro-1H-indol-4(5H)-one O...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of hERG expressed in HEK cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194358((E)--2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-phe...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of hERG expressed in HEK cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed