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Found 136 Enz. Inhib. hit(s) with all data for entry = 50018511
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196560((2R,3R,4S,5R)-2-(6-(bicyclo[2.2.1]heptan-1-ylamino...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196555(1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196557(1-(6-(cyclopentylamino)-9-((2R,3R,4S,5R)-3,4-dihyd...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196558(1-(6-(p-toluidino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196563(CHEMBL392958 | ethyl 1-(6-(cyclopentylamino)-9-((2...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196543(1-(6-(bicyclo[2.2.1]heptan-1-ylamino)-9-((2R,3R,4S...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196541(1-(6-(cyclopentylamino)-9-((2R,3R,4S,5R)-3,4-dihyd...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196546(1-(6-(cyclopentylamino)-9-((2R,3R,4S,5R)-3,4-dihyd...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196569(CHEMBL232516 | N-benzyl-1-(9-((2R,3R,4S,5R)-3,4-di...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196564((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(methylamino)...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196566(CHEMBL234974 | ethyl 1-(6-(bicyclo[2.2.1]heptan-1-...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196552(CHEMBL398588 | ethyl 1-(9-((2R,3R,4S,5R)-3,4-dihyd...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196540((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxyme...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196548(CHEMBL231881 | N-(4-chlorobenzyl)-1-(9-((2R,3R,4S,...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196561((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxyme...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196553(CHEMBL393295 | ethyl 4-((1-(9-((2R,3R,4S,5R)-3,4-d...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196565(1-(6-(cyclohexylamino)-9-((2R,3R,4S,5R)-3,4-dihydr...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196542(4-((1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxyme...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196556(1-(6-(cyclopentylamino)-9-((2R,3R,4S,5R)-3,4-dihyd...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196570(1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196572(1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196550((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(4-methoxy...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196547((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxyme...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196573(CHEMBL234779 | N-(4-fluorobenzyl)-1-(9-((2R,3R,4S,...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196563(CHEMBL392958 | ethyl 1-(6-(cyclopentylamino)-9-((2...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196538((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxyme...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196541(1-(6-(cyclopentylamino)-9-((2R,3R,4S,5R)-3,4-dihyd...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196545(1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196559(1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196571((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxyme...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196548(CHEMBL231881 | N-(4-chlorobenzyl)-1-(9-((2R,3R,4S,...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196554(CHEMBL428716 | ethyl 1-(6-(cyclohexylamino)-9-((2R...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196554(CHEMBL428716 | ethyl 1-(6-(cyclohexylamino)-9-((2R...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196547((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxyme...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196549((2R,3R,4S,5R)-2-(6-(cyclopentylamino)-2-(1H-pyrazo...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196538((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxyme...)
Affinity DataKi:  36nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196540((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxyme...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196571((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxyme...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196552(CHEMBL398588 | ethyl 1-(9-((2R,3R,4S,5R)-3,4-dihyd...)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196568((2R,3R,4S,5R)-2-(6-(ethylamino)-2-(4-(4-methoxyphe...)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196573(CHEMBL234779 | N-(4-fluorobenzyl)-1-(9-((2R,3R,4S,...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196570(1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196569(CHEMBL232516 | N-benzyl-1-(9-((2R,3R,4S,5R)-3,4-di...)
Affinity DataKi:  54nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196544((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(2-(4-(hydroxyme...)
Affinity DataKi:  63nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196562(2-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196567(1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  73nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196551((2R,3R,4S,5R)-2-(6-(p-toluidino)-2-(4-(hydroxymeth...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196562(2-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  77nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196555(1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl...)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in DDT membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50196553(CHEMBL393295 | ethyl 4-((1-(9-((2R,3R,4S,5R)-3,4-d...)
Affinity DataKi:  92nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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