Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50018698
TargetTransporter(Rattus norvegicus)
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198230((S)-2-((S)-(2-iodophenoxy)(phenyl)methyl)morpholin...)
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198226(2-((2-iodophenoxy)(phenyl)methyl)morpholine | CHEM...)
Affinity DataKi:  2.47nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198231(2-((2-nitrobenzyloxy)(3-iodophenyl)methyl)morpholi...)
Affinity DataKi:  14.2nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198233(2-((3-iodophenyl)(2-methoxyphenoxy)methyl)morpholi...)
Affinity DataKi:  15.4nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198232(2-((3-iodophenyl)(o-tolyloxy)methyl)morpholine | C...)
Affinity DataKi:  27.6nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198227(2-((2-ethoxyphenoxy)(3-iodophenyl)methyl)morpholin...)
Affinity DataKi:  28.5nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198230((S)-2-((S)-(2-iodophenoxy)(phenyl)methyl)morpholin...)
Affinity DataKi:  40.4nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198231(2-((2-nitrobenzyloxy)(3-iodophenyl)methyl)morpholi...)
Affinity DataKi:  70.4nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198234(2-((5-iodothiophen-2-yl)(o-tolyloxy)methyl)morphol...)
Affinity DataKi:  71.9nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198225(2-((2-methoxybenzyloxy)(3-iodophenyl)methyl)morpho...)
Affinity DataKi:  73.8nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198228(2-((5-iodothiophen-2-yl)(2-methoxyphenoxy)methyl)m...)
Affinity DataKi:  79.6nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198229(2-((3-iodophenyl)(2-(trifluoromethyl)phenoxy)methy...)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198228(2-((5-iodothiophen-2-yl)(2-methoxyphenoxy)methyl)m...)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198234(2-((5-iodothiophen-2-yl)(o-tolyloxy)methyl)morphol...)
Affinity DataKi:  186nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198228(2-((5-iodothiophen-2-yl)(2-methoxyphenoxy)methyl)m...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198230((S)-2-((S)-(2-iodophenoxy)(phenyl)methyl)morpholin...)
Affinity DataKi:  228nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198231(2-((2-nitrobenzyloxy)(3-iodophenyl)methyl)morpholi...)
Affinity DataKi:  252nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198225(2-((2-methoxybenzyloxy)(3-iodophenyl)methyl)morpho...)
Affinity DataKi:  351nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198226(2-((2-iodophenoxy)(phenyl)methyl)morpholine | CHEM...)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198229(2-((3-iodophenyl)(2-(trifluoromethyl)phenoxy)methy...)
Affinity DataKi:  486nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198225(2-((2-methoxybenzyloxy)(3-iodophenyl)methyl)morpho...)
Affinity DataKi:  716nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198232(2-((3-iodophenyl)(o-tolyloxy)methyl)morpholine | C...)
Affinity DataKi:  740nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198229(2-((3-iodophenyl)(2-(trifluoromethyl)phenoxy)methy...)
Affinity DataKi:  1.87E+3nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198227(2-((2-ethoxyphenoxy)(3-iodophenyl)methyl)morpholin...)
Affinity DataKi:  3.14E+3nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases

Curated by ChEMBL
LigandPNGBDBM50198233(2-((3-iodophenyl)(2-methoxyphenoxy)methyl)morpholi...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed