Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50000624
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007965(CHEMBL312194 | Tyr(psi)CH2O-Gly-Gly-Phe-Leu-NH2 | ...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity of the compound to opioid receptor mu was determined in rat brain using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity of the compound to opioid receptor mu was determined in rat brain using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007965(CHEMBL312194 | Tyr(psi)CH2O-Gly-Gly-Phe-Leu-NH2 | ...)
Affinity DataKi:  7.80nMAssay Description:Binding affinity of the compound to opioid receptor delta was determined in rat brain using [3H]-DSTBULET as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  629nMAssay Description:Binding affinity of the compound to opioid receptor delta was determined in rat brain using [3H]-DSTBULET as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007966(CHEMBL420022 | Tyr-Gly(psi)CH2O-Gly-PheLeu-NH2)
Affinity DataKi:  1.38E+3nMAssay Description:Binding affinity of the compound to opioid receptor mu was determined in rat brain using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007966(CHEMBL420022 | Tyr-Gly(psi)CH2O-Gly-PheLeu-NH2)
Affinity DataKi:  9.20E+3nMAssay Description:Binding affinity of the compound to opioid receptor delta was determined in rat brain using [3H]-DSTBULET as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007972(CHEMBL311917 | pGlu6-Phe-Phe8(psi)CH2O-Gly-Leu-Met...)
Affinity DataEC50:  40nMAssay Description:Effective dose of the compound was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007963(CHEMBL441061 | pGlu6-Phe-Phe-Gly-Leu-Met-NH2)
Affinity DataEC50:  2.20nMAssay Description:Effective dose of the compound was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007963(CHEMBL441061 | pGlu6-Phe-Phe-Gly-Leu-Met-NH2)
Affinity DataEC50:  5nMAssay Description:Effective dose of the compound was measured on NK3 receptors of guinea pig ileum for maximal contraction in the presence of 10e-7 M substance P methy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007972(CHEMBL311917 | pGlu6-Phe-Phe8(psi)CH2O-Gly-Leu-Met...)
Affinity DataEC50:  13nMAssay Description:Effective dose of the compound was measured on NK3 receptors of guinea pig ileum for maximal contraction in the presence of 10e-7 M substance P methy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007962(CHEMBL81919 | pGlu6-Phe-NMePhe-Gly-Leu-Met-NH2)
Affinity DataEC50:  0.900nMAssay Description:Effective dose of the compound was measured on NK3 receptors of guinea pig ileum for maximal contraction in the presence of 10e-7 M substance P methy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007962(CHEMBL81919 | pGlu6-Phe-NMePhe-Gly-Leu-Met-NH2)
Affinity DataEC50:  600nMAssay Description:Effective dose of the compound was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed