Compile Data Set for Download or QSAR
maximum 50k data
Found 60 Enz. Inhib. hit(s) with all data for entry = 50019602
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206043(((2S,4S)-4-(4-(5-nitropyridin-2-yl)piperazin-1-yl)...)
Affinity DataIC50:  0.920nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206058(6-(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidi...)
Affinity DataIC50:  1nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206043(((2S,4S)-4-(4-(5-nitropyridin-2-yl)piperazin-1-yl)...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206047(2-(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidi...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206047(2-(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidi...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206032(4-(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidi...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206058(6-(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidi...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206037(CHEMBL241252 | thiazolidin-3-yl((2S,4S)-4-(4-(5-(t...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206040(2-(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidi...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206038(((2S,4S)-4-(4-(4-nitrophenyl)piperazin-1-yl)pyrrol...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206032(4-(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidi...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206037(CHEMBL241252 | thiazolidin-3-yl((2S,4S)-4-(4-(5-(t...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206040(2-(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidi...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206038(((2S,4S)-4-(4-(4-nitrophenyl)piperazin-1-yl)pyrrol...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206054(((2S,4S)-4-(4-(4-nitrophenyl)piperidin-1-yl)pyrrol...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206044(((2S,4S)-4-(4-(4-nitrophenyl)-1,4-diazepan-1-yl)py...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206059(((2S,4S)-4-(4-(5-chloropyridin-2-yl)piperazin-1-yl...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206052(((2S,4S)-4-(4-(pyridin-2-yl)piperazin-1-yl)pyrroli...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206044(((2S,4S)-4-(4-(4-nitrophenyl)-1,4-diazepan-1-yl)py...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206031(((2S,4S)-4-(4-(3,4-dichlorophenyl)piperazin-1-yl)p...)
Affinity DataIC50:  3nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206057(((2S,4S)-4-(4-(pyridin-4-yl)piperazin-1-yl)pyrroli...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206059(((2S,4S)-4-(4-(5-chloropyridin-2-yl)piperazin-1-yl...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206054(((2S,4S)-4-(4-(4-nitrophenyl)piperidin-1-yl)pyrrol...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206052(((2S,4S)-4-(4-(pyridin-2-yl)piperazin-1-yl)pyrroli...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206057(((2S,4S)-4-(4-(pyridin-4-yl)piperazin-1-yl)pyrroli...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206050(((2S,4S)-4-(4-(3-chlorophenyl)piperazin-1-yl)pyrro...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206031(((2S,4S)-4-(4-(3,4-dichlorophenyl)piperazin-1-yl)p...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206046(4-(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidi...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206046(4-(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidi...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206053(((2S,4S)-4-(4-phenylpiperidin-1-yl)pyrrolidin-2-yl...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206048(CHEMBL241245 | thiazolidin-3-yl((2S,4S)-4-(4-(4-(t...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206048(CHEMBL241245 | thiazolidin-3-yl((2S,4S)-4-(4-(4-(t...)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206050(((2S,4S)-4-(4-(3-chlorophenyl)piperazin-1-yl)pyrro...)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206036(((2S,4S)-4-(4-(4-bromophenyl)piperazin-1-yl)pyrrol...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206039(((2S,4S)-4-(4-(4-chlorophenyl)piperazin-1-yl)pyrro...)
Affinity DataIC50:  8.70nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206036(((2S,4S)-4-(4-(4-bromophenyl)piperazin-1-yl)pyrrol...)
Affinity DataIC50:  9nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206053(((2S,4S)-4-(4-phenylpiperidin-1-yl)pyrrolidin-2-yl...)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206039(((2S,4S)-4-(4-(4-chlorophenyl)piperazin-1-yl)pyrro...)
Affinity DataIC50:  10.3nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206055(((2S,4S)-4-(4-(2-chlorophenyl)piperazin-1-yl)pyrro...)
Affinity DataIC50:  10.8nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206056(((2S,4S)-4-(4-phenylpiperazin-1-yl)pyrrolidin-2-yl...)
Affinity DataIC50:  10.9nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206055(((2S,4S)-4-(4-(2-chlorophenyl)piperazin-1-yl)pyrro...)
Affinity DataIC50:  10.9nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206041(((2S,4S)-4-(4-(4-fluorophenyl)piperazin-1-yl)pyrro...)
Affinity DataIC50:  12.2nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206051(((2S,4S)-4-(4-(4-methoxyphenyl)piperazin-1-yl)pyrr...)
Affinity DataIC50:  13.5nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206035(((2S,4S)-4-morpholinopyrrolidin-2-yl)(thiazolidin-...)
Affinity DataIC50:  13.9nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206051(((2S,4S)-4-(4-(4-methoxyphenyl)piperazin-1-yl)pyrr...)
Affinity DataIC50:  16.9nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206041(((2S,4S)-4-(4-(4-fluorophenyl)piperazin-1-yl)pyrro...)
Affinity DataIC50:  17.5nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206056(((2S,4S)-4-(4-phenylpiperazin-1-yl)pyrrolidin-2-yl...)
Affinity DataIC50:  17.6nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206035(((2S,4S)-4-morpholinopyrrolidin-2-yl)(thiazolidin-...)
Affinity DataIC50:  18.9nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206034(((2S,4S)-4-(4-benzhydrylpiperazin-1-yl)pyrrolidin-...)
Affinity DataIC50:  21nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50206049(((2S,4S)-4-(4-benzylpiperazin-1-yl)pyrrolidin-2-yl...)
Affinity DataIC50:  30.5nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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