Compile Data Set for Download or QSAR
maximum 50k data
Found 46 Enz. Inhib. hit(s) with all data for entry = 50035989
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKi:  1.40nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKi:  1.90nMAssay Description:Inhibition of the 3 nM VP stimulation of phospholipase-C in cultured WRK cells was used as a V1-mediated assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008092(CHEMBL2372415 | cyclo(Ppa-Phe(NO2)-Phe-Val-Asn-Cys...)
Affinity DataKd:  3.20nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKd:  0.479nMAssay Description:Negative log of Kd.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008096(CHEMBL2372414 | cyclo(Ppa-Phe(N3)-Phe-Val-Asn-Cys)...)
Affinity DataKd:  35nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008084(1-[13-Benzyl-7-carbamoylmethyl-10-isopropyl-16-(4-...)
Affinity DataKd:  41nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008088(CHEMBL2372416 | cyclo(Depa-Phe(N3)-Phe-Val-Asn-Cys...)
Affinity DataKd:  2.60nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008083(CHEMBL2372418 | [2-({1-[19-Amino-10-(2-carbamoyl-e...)
Affinity DataKd:  54nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008085(CHEMBL2028984 | [2-({1-[19-Amino-13-(4-azido-benzy...)
Affinity DataKd:  76nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453152(CHEMBL2115365)
Affinity DataKd:  2.63nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453150(CHEMBL2372420)
Affinity DataKd:  27nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453151(CHEMBL2372421)
Affinity DataKd:  33nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453148(CHEMBL2372422)
Affinity DataKd:  16nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008091(1-[16-(4-Azido-benzyl)-13-benzyl-7-carbamoylmethyl...)
Affinity DataKd:  5nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Sus scrofa)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKd:  100nMAssay Description:Binding affinity towards V2-receptor in LLCPK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Sus scrofa)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKd:  100nMAssay Description:Binding affinity towards Vasopressin V2 receptor in LLCPK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKd:  0.182nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008097(CHEMBL2028983 | [2-({1-[19-Amino-13-(4-azido-benzy...)
Affinity DataKd:  0.331nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453149(CHEMBL2115368)
Affinity DataKd:  1.80nMAssay Description:Binding potency against V1 receptor in rat liver cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453149(CHEMBL2115368)
Affinity DataKd:  1.80nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKd:  0.480nMAssay Description:Inhibition of the 3 nM VP stimulation of phospholipase-C in cultured WRK cells was used as a V1-mediated assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008083(CHEMBL2372418 | [2-({1-[19-Amino-10-(2-carbamoyl-e...)
Affinity DataKd:  54nMAssay Description:Inhibition of the 3 nM VP stimulation of phospholipase-C in cultured WRK cells was used as a V1-mediated assay (Vasopressin V1 receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008091(1-[16-(4-Azido-benzyl)-13-benzyl-7-carbamoylmethyl...)
Affinity DataKd:  4.90nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453150(CHEMBL2372420)
Affinity DataKd:  27nMAssay Description:Negative log of Kd.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453151(CHEMBL2372421)
Affinity DataKd:  33nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008088(CHEMBL2372416 | cyclo(Depa-Phe(N3)-Phe-Val-Asn-Cys...)
Affinity DataKd:  2.60nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453148(CHEMBL2372422)
Affinity DataKd:  16nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008084(1-[13-Benzyl-7-carbamoylmethyl-10-isopropyl-16-(4-...)
Affinity DataKd:  41nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKd:  0.646nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008096(CHEMBL2372414 | cyclo(Ppa-Phe(N3)-Phe-Val-Asn-Cys)...)
Affinity DataKd:  36nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008092(CHEMBL2372415 | cyclo(Ppa-Phe(NO2)-Phe-Val-Asn-Cys...)
Affinity DataKd:  3.20nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKd:  0.180nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKd:  0.180nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008097(CHEMBL2028983 | [2-({1-[19-Amino-13-(4-azido-benzy...)
Affinity DataKd:  0.330nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008097(CHEMBL2028983 | [2-({1-[19-Amino-13-(4-azido-benzy...)
Affinity DataKd:  0.330nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008085(CHEMBL2028984 | [2-({1-[19-Amino-13-(4-azido-benzy...)
Affinity DataKd:  75nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453149(CHEMBL2115368)
Affinity DataKd:  1.70nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKd:  0.600nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453152(CHEMBL2115365)
Affinity DataKd:  2.60nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKd:  0.603nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453152(CHEMBL2115365)
Affinity DataKd:  2.60nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453152(CHEMBL2115365)
Affinity DataKd:  2.64nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50008097(CHEMBL2028983 | [2-({1-[19-Amino-13-(4-azido-benzy...)
Affinity DataKd:  0.331nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50453149(CHEMBL2115368)
Affinity DataKd:  1.80nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKd:  0.640nMAssay Description:Binding potency against V1 receptor in rat liver cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKd:  0.182nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed