Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50037875
TargetDelta-type opioid receptor(MOUSE)
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]NTI from delta opioid receptor in CD1 mouse brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209644(17-cyclopropylmethyl)-6,7-didehydro-4,5alpha-epoxy...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]NTI from delta opioid receptor in CD1 mouse brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209645(17-(cyclopropylmethyl)-6,7-didehydro-4,5alpha-epox...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]NTI from delta opioid receptor in CD1 mouse brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  14.9nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209644(17-cyclopropylmethyl)-6,7-didehydro-4,5alpha-epoxy...)
Affinity DataKi:  26.2nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  33.9nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209644(17-cyclopropylmethyl)-6,7-didehydro-4,5alpha-epoxy...)
Affinity DataKi:  48.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209645(17-(cyclopropylmethyl)-6,7-didehydro-4,5alpha-epox...)
Affinity DataKi:  1.75E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209645(17-(cyclopropylmethyl)-6,7-didehydro-4,5alpha-epox...)
Affinity DataKi:  2.01E+3nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed