Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50025233
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50220067(11H-2,5,11-triaza-benzo[a]trindene-1,3,4,6-tetraon...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50236805(4,5-dihydro-11H-2,5,11-triaza-benzo[a]trindene-1,3...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50216165(1,11-dihydro-1,3,5,11-tetraaza-benzo[a]trindene-4,...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50251213(6H-2-N-hydroxymethyl-5-ethoxycarbonyl-pyrrolo-[3,4...)
Affinity DataIC50:  210nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50251201(6,11-Dihydro-5H-2,5,11-triaza-benzo[a]trindene-1,3...)
Affinity DataIC50:  370nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50216157(11H-2,5,11,11b-Tetraaza-benzo[a]trindene-4,6-dione...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50251206(2H,6H-5-Ethoxycarbonyl-1,3-dihydropyrrolo-[3,4-c]c...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed