Compile Data Set for Download or QSAR
maximum 50k data
Found 43 Enz. Inhib. hit(s) with all data for entry = 2928
LigandPNGBDBM26166(2,4-dianilino pyrimidine, 23 | 3-({4-[(5-hydroxy-2...)
Affinity DataIC50:  8.5nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26180(2,4-dianilino pyrimidine, 37 | 3-({4-[(5-methyl-1H...)
Affinity DataIC50:  12nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26145(2,4-dianilino pyrimidine, 2 | 3-({4-[(5-hydroxy-2-...)
Affinity DataIC50:  13nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26186(2,4-dianilino pyrimidine, 43 | 3-({4-[(5-methyl-1H...)
Affinity DataIC50:  19nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26185(2,4-dianilino pyrimidine, 42 | 3-{[4-(1H-indazol-4...)
Affinity DataIC50:  33nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26152(2,4-dianilino pyrimidine, 9 | 3-({4-[(4-hydroxy-2-...)
Affinity DataIC50:  40nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26149(2,4-dianilino pyrimidine, 6 | 3-({4-[(2-bromo-5-hy...)
Affinity DataIC50:  41nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26167(2,4-dianilino pyrimidine, 24 | 3-({4-[(5-methoxy-2...)
Affinity DataIC50:  54nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26182(2,4-dianilino pyrimidine, 39 | 3-({4-[(7-methyl-1H...)
Affinity DataIC50:  55nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25191(4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-y...)
Affinity DataIC50:  59nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26147(2,4-dianilino pyrimidine, 4 | 3-({4-[(3-hydroxy-5-...)
Affinity DataIC50:  73nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26156(2,4-dianilino pyrimidine, 13 | 3-({4-[(5-methoxy-2...)
Affinity DataIC50:  86nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26151(2,4-dianilino pyrimidine, 8 | 3-({4-[(2-methylphen...)
Affinity DataIC50:  89nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26157(2,4-dianilino pyrimidine, 14 | 3-({4-[(5-amino-2-m...)
Affinity DataIC50:  97nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26153(2,4-dianilino pyrimidine, 10 | 3-({4-[(2-hydroxy-6...)
Affinity DataIC50:  100nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26179(2,4-dianilino pyrimidine, 36 | 3-{[4-(1H-indazol-4...)
Affinity DataIC50:  100nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26146(2,4-dianilino pyrimidine, 3 | 3-({4-[(3-hydroxyphe...)
Affinity DataIC50:  130nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26148(2,4-dianilino pyrimidine, 5 | 3-({4-[(3-hydroxy-4-...)
Affinity DataIC50:  190nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26154(2,4-dianilino pyrimidine, 11 | 3-({4-[(5-fluoro-2-...)
Affinity DataIC50:  270nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26168(2,4-dianilino pyrimidine, 25 | 3-({4-[(2,4-difluor...)
Affinity DataIC50:  350nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM26155(2,4-dianilino pyrimidine, 12 | 3-({4-[(5-chloro-2-...)
Affinity DataIC50:  380nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26176(2,4-dianilino pyrimidine, 33 | 3-{[4-(1H-1,2,3-ben...)
Affinity DataIC50:  490nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26181(2,4-dianilino pyrimidine, 38 | 3-({4-[(6-methyl-1H...)
Affinity DataIC50:  520nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26175(2,4-dianilino pyrimidine, 32 | 3-{[4-(quinolin-5-y...)
Affinity DataIC50:  560nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM26150(2,4-dianilino pyrimidine, 7 | 3-[(4-{[5-hydroxy-2-...)
Affinity DataIC50:  880nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26165(2,4-dianilino pyrimidine, 22 | 3-({4-[(2,4-difluor...)
Affinity DataIC50:  1.10E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26158(2,4-dianilino pyrimidine, 15 | 3-({2-[(3-carbamoyl...)
Affinity DataIC50:  1.30E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26177(2,4-dianilino pyrimidine, 34 | 3-{[4-(1H-indazol-7...)
Affinity DataIC50:  1.40E+3nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26183(2,4-dianilino pyrimidine, 40 | 3-({4-[(1-methyl-1H...)
Affinity DataIC50:  1.60E+3nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26172(2,4-dianilino pyrimidine, 29 | 3-({4-[(1-methyl-1H...)
Affinity DataIC50:  1.80E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26164(2,4-dianilino pyrimidine, 21 | 3-[(4-{[3-(N-methyl...)
Affinity DataIC50:  1.80E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM26162(2,4-dianilino pyrimidine, 19 | 3-({4-[(3-methoxyph...)
Affinity DataIC50:  2.70E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26184(2,4-dianilino pyrimidine, 41 | 3-({4-[(1,5-dimethy...)
Affinity DataIC50:  2.80E+3nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26169(2,4-dianilino pyrimidine, 26 | 3-{[4-(1,3-benzothi...)
Affinity DataIC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM26171(2,4-dianilino pyrimidine, 28 | 3-{[4-(1H-indazol-5...)
Affinity DataIC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26163(2,4-dianilino pyrimidine, 20 | 3-({4-[(3-fluorophe...)
Affinity DataIC50:  3.30E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26161(2,4-dianilino pyrimidine, 18 | 3-[(4-{[5-(aminomet...)
Affinity DataIC50:  3.40E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26173(2,4-dianilino pyrimidine, 30 | 3-{[4-(1H-1,2,3-ben...)
Affinity DataIC50:  4.40E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26178(2,4-dianilino pyrimidine, 35 | 3-({4-[(2-methyl-1H...)
Affinity DataIC50:  5.60E+3nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM26160(2,4-dianilino pyrimidine, 17 | 3-({4-[(5-methanesu...)
Affinity DataIC50:  7.70E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM26174(2,4-dianilino pyrimidine, 31 | 3-({4-[(1-methyl-1H...)
Affinity DataIC50:  8.20E+3nMAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26159(2,4-dianilino pyrimidine, 16 | 3-({2-[(3-carbamoyl...)
Affinity DataIC50:  9.30E+3nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM26170(2,4-dianilino pyrimidine, 27 | 3-({4-[(1-methyl-1H...)
Affinity DataIC50:  1.60E+4nMpH: 7.4 T: 2°CAssay Description:Lck activity was assessed using a TR-FRET assay in a 384-well plate format. The degree of phosphorylation of Biotinylated substrate was measured usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed