Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50021543
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50198419(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  16nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225715(3-(3,5-bis(trifluoromethyl)phenyl)-1-(1-(((1R,5S)-...)
Affinity DataKi:  26nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225718(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  100nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225729(3-(4-chloro-3-(trifluoromethyl)phenyl)-1-(1-(((1R,...)
Affinity DataKi:  120nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225725(6-bromo-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]h...)
Affinity DataKi:  130nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225711(CHEMBL437776 | N-(1-(((1R,5S)-6,6-dimethylbicyclo[...)
Affinity DataKi:  140nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225726(4-bromo-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]h...)
Affinity DataKi:  150nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225731(1-(3,5-bis(trifluoromethyl)phenyl)-3-(1-(((1R,5S)-...)
Affinity DataKi:  170nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225733(6-chloro-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]...)
Affinity DataKi:  170nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225732(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  180nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225714(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  200nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225710(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  220nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225724(CHEMBL250658 | N-(4-(3,5-bis(trifluoromethyl)pheny...)
Affinity DataKi:  260nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225728(CHEMBL250483 | N-(3-(3,5-bis(trifluoromethyl)pheny...)
Affinity DataKi:  270nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225722(5-chloro-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]...)
Affinity DataKi:  290nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225717(CHEMBL249016 | N-(1-(((1R,5S)-6,6-dimethylbicyclo[...)
Affinity DataKi:  350nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225716(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  380nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225720(CHEMBL250657 | N-(4-(3,4-dichlorophenyl)thiazol-2-...)
Affinity DataKi:  460nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225712(4-chloro-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]...)
Affinity DataKi:  460nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225721(7-chloro-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]...)
Affinity DataKi:  620nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225709(CHEMBL249612 | N-(1-(((1R,5S)-6,6-dimethylbicyclo[...)
Affinity DataKi:  680nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225723(CHEMBL249014 | N-(1-(((1R,5S)-6,6-dimethylbicyclo[...)
Affinity DataKi:  720nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225719(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  750nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225734(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-...)
Affinity DataKi:  880nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225727(CHEMBL248632 | N-(1-(((1R,5S)-6,6-dimethylbicyclo[...)
Affinity DataKi:  950nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225730(3-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  3.50E+3nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50225713(1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...)
Affinity DataKi:  3.60E+3nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed