Compile Data Set for Download or QSAR
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Found 16 Enz. Inhib. hit(s) with all data for entry = 50021647
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226429(CHEMBL237354 | [L-arginyl]-N-(2,4-dichlorophenethy...)
Affinity DataIC50:  170nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226436(CHEMBL401228 | [L-arginyl]-[N-(2,4-dichloropheneth...)
Affinity DataIC50:  180nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226431(CHEMBL237138 | [[N-(2,4-dichlorophenethyl)-N-(6-am...)
Affinity DataIC50:  400nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226430(CHEMBL400008 | [L-arginyl]-[N-[2-(indol-3-yl)ethyl...)
Affinity DataIC50:  520nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226432(CHEMBL430173 | cis-(L-arginyl)amino-N-(2,4-dichlor...)
Affinity DataIC50:  700nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226435((S)-N-(2,4-dichlorophenethyl)-N-(2-((2,4-dichlorop...)
Affinity DataIC50:  700nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226429(CHEMBL237354 | [L-arginyl]-N-(2,4-dichlorophenethy...)
Affinity DataIC50:  800nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226434(CHEMBL392540 | [L-arginyl]-N-[2-(indol-3-yl)ethyl]...)
Affinity DataIC50:  1.10E+3nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226433(CHEMBL395124 | [L-arginyl]-[N-[2-(indol-3-yl)-ethy...)
Affinity DataIC50:  1.33E+3nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226431(CHEMBL237138 | [[N-(2,4-dichlorophenethyl)-N-(6-am...)
Affinity DataIC50:  3.00E+3nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226432(CHEMBL430173 | cis-(L-arginyl)amino-N-(2,4-dichlor...)
Affinity DataIC50:  8.00E+3nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226435((S)-N-(2,4-dichlorophenethyl)-N-(2-((2,4-dichlorop...)
Affinity DataIC50:  1.50E+4nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226430(CHEMBL400008 | [L-arginyl]-[N-[2-(indol-3-yl)ethyl...)
Affinity DataIC50:  1.70E+4nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226434(CHEMBL392540 | [L-arginyl]-N-[2-(indol-3-yl)ethyl]...)
Affinity DataIC50:  1.80E+4nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226436(CHEMBL401228 | [L-arginyl]-[N-(2,4-dichloropheneth...)
Affinity DataIC50:  1.66E+5nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226433(CHEMBL395124 | [L-arginyl]-[N-[2-(indol-3-yl)-ethy...)
Affinity DataIC50:  2.07E+5nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed