Affinity DataKi: 19.5nMAssay Description:Displacement of [125I]ABMECA from human adenosine A3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 25.3nMAssay Description:Displacement of [125I]ABMECA from human adenosine A3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 26.7nMAssay Description:Displacement of [125I]ABMECA from human adenosine A3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 27.2nMAssay Description:Displacement of [125I]ABMECA from human adenosine A3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [125I]ABMECA from human adenosine A3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 87.5nMAssay Description:Displacement of [125I]ABMECA from human adenosine A3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 98.3nMAssay Description:Displacement of [125I]ABMECA from human adenosine A3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 182nMAssay Description:Displacement of [125I]ABMECA from human adenosine A3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Displacement of [125I]ABMECA from human adenosine A3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Displacement of [125I]ABMECA from human adenosine A3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 125nMAssay Description:Activity at human adenosine A3 receptor expressed in CHO cells assessed as antagonism of Cl-IB-MECA-inhibited cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Activity at human adenosine A3 receptor expressed in CHO cells assessed as antagonism of Cl-IB-MECA-inhibited cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 238nMAssay Description:Activity at human adenosine A3 receptor expressed in CHO cells assessed as antagonism of Cl-IB-MECA-inhibited cAMP productionMore data for this Ligand-Target Pair