Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50022194
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Molsoft

Curated by ChEMBL
LigandPNGBDBM50232469(CHEMBL252145 | N,N-bis(tosylmethyl)hexan-1-amine)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Molsoft

Curated by ChEMBL
LigandPNGBDBM50232467(CHEMBL399303 | phenyl-N,N-bis(tosylmethyl)methanam...)
Affinity DataKi:  7.50E+3nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Molsoft

Curated by ChEMBL
LigandPNGBDBM50232470(2-phenyl-N,N-bis(o-tolylthiomethyl)ethanamine | CH...)
Affinity DataKi:  7.50E+3nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Molsoft

Curated by ChEMBL
LigandPNGBDBM50232468(6-(((3-chlorobenzyl)(methyl)amino)methyl)-N2-o-tol...)
Affinity DataKi:  7.80E+3nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Molsoft

Curated by ChEMBL
LigandPNGBDBM50232466(2-(dimethylamino)ethyl 4-(5-(4-methoxybenzylidene)...)
Affinity DataKi:  8.10E+3nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Molsoft

Curated by ChEMBL
LigandPNGBDBM50232465(4-methoxy-benzoic acid 2-diethylaminomethyl-4-(1,1...)
Affinity DataKi:  1.13E+4nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Molsoft

Curated by ChEMBL
LigandPNGBDBM50232464(CHEMBL251947 | {3-[2-(4-bromo-phenyl)-benzo[d]imid...)
Affinity DataKi:  1.19E+4nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Molsoft

Curated by ChEMBL
LigandPNGBDBM50232471(CHEMBL251948 | N-(3-(benzyl(isopropyl)amino)propyl...)
Affinity DataKi:  2.09E+4nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed