Compile Data Set for Download or QSAR
maximum 50k data
Found 82 Enz. Inhib. hit(s) with all data for entry = 50022295
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233576((R)-3-(2-(1-(4-bromofuran-2-yl)propylamino)-3,4-di...)
Affinity DataIC50:  2nMAssay Description:Inhibition of CXCR2-mediated chemotaxis in Ba/F3 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233586(2-hydroxy-3-(2-(1-(5-(hydroxymethyl)furan-2-yl)pro...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233554((R)-3-(3,4-dioxo-2-(1-(pyridin-2-yl)propylamino)cy...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233561((R)-3-(3,4-dioxo-2-(1-(thiophen-3-yl)propylamino)c...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233576((R)-3-(2-(1-(4-bromofuran-2-yl)propylamino)-3,4-di...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233560(3-(2-(1-(benzofuran-2-yl)propylamino)-3,4-dioxocyc...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233574((R)-3-(2-(1-(4-chlorofuran-2-yl)propylamino)-3,4-d...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233592(3-(2-(1-(5-ethylfuran-2-yl)propylamino)-3,4-dioxoc...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233554((R)-3-(3,4-dioxo-2-(1-(pyridin-2-yl)propylamino)cy...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of CXCR2-mediated chemotaxis in Ba/F3 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233589(3-(2-(1-(4-chlorofuran-2-yl)propylamino)-3,4-dioxo...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233572((R)-3-(2-(1-(5-chlorofuran-2-yl)propylamino)-3,4-d...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233588(3-(2-(1-(5-bromofuran-2-yl)propylamino)-3,4-dioxoc...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233581(3-(2-(1-(5-chlorofuran-2-yl)propylamino)-3,4-dioxo...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233563(3-(2-(1-(furan-2-yl)propylamino)-3,4-dioxocyclobut...)
Affinity DataIC50:  5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233577(3-(2-(1-(4-bromofuran-2-yl)propylamino)-3,4-dioxoc...)
Affinity DataIC50:  5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233553(2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylfuran-2-yl...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233584(3-(3,4-dioxo-2-(1-(thiophen-3-yl)propylamino)cyclo...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233570(3-(3,4-dioxo-2-(1-(4-phenylfuran-2-yl)propylamino)...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233580(3-(3,4-dioxo-2-(1-(thiophen-2-yl)propylamino)cyclo...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233557(3-(2-(1-(5-chlorothiophen-2-yl)propylamino)-3,4-di...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233558((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylisoxaz...)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233568(3-(2-(1-(5-(difluoromethyl)furan-2-yl)propylamino)...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233567(2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylisoxazol-3...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233590(3-(2-(1-(4-(3,5-dimethylisoxazol-4-yl)furan-2-yl)p...)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233552(3-(2-(1-(furan-3-yl)propylamino)-3,4-dioxocyclobut...)
Affinity DataIC50:  8nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233562(3-(3,4-dioxo-2-(1-(4-(thiophen-3-yl)furan-2-yl)pro...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233556(2-hydroxy-N,N-dimethyl-3-(2-(1-(3-methyl-1,2,4-oxa...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233565(2-hydroxy-N,N-dimethyl-3-(2-(1-(oxazol-2-yl)propyl...)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233587(3-(3,4-dioxo-2-(1-(4-(pyridin-4-yl)furan-2-yl)prop...)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233583(3-(3,4-dioxo-2-(1-(thiazol-2-yl)propylamino)cyclob...)
Affinity DataIC50:  9.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233578(2-hydroxy-3-(2-(1-(isoxazol-5-yl)propylamino)-3,4-...)
Affinity DataIC50:  9.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233569(2-hydroxy-N,N-dimethyl-3-(2-(1-(oxazol-4-yl)propyl...)
Affinity DataIC50:  10.9nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233558((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylisoxaz...)
Affinity DataIC50:  12.2nMAssay Description:Inhibition of CXCR2-mediated chemotaxis in Ba/F3 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233579(3-(2-(1-(3-bromofuran-2-yl)propylamino)-3,4-dioxoc...)
Affinity DataIC50:  16.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233566(3-(3,4-dioxo-2-(1-(5-(trifluoromethyl)furan-2-yl)p...)
Affinity DataIC50:  17.2nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233564(3-(2-(1-(3-chlorothiophen-2-yl)propylamino)-3,4-di...)
Affinity DataIC50:  21nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233591(3-(2-(1-(5-(2-chlorophenyl)furan-2-yl)propylamino)...)
Affinity DataIC50:  49nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233555(3-(3,4-dioxo-2-(1-(pyridin-4-yl)propylamino)cyclob...)
Affinity DataIC50:  50nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233576((R)-3-(2-(1-(4-bromofuran-2-yl)propylamino)-3,4-di...)
Affinity DataIC50:  55nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233573(3-(2-(1-(5-(3-chlorophenyl)furan-2-yl)propylamino)...)
Affinity DataIC50:  58nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233574((R)-3-(2-(1-(4-chlorofuran-2-yl)propylamino)-3,4-d...)
Affinity DataIC50:  62nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233563(3-(2-(1-(furan-2-yl)propylamino)-3,4-dioxocyclobut...)
Affinity DataIC50:  67nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233582(3-(3,4-dioxo-2-(1-(5-(3-(trifluoromethyl)phenyl)fu...)
Affinity DataIC50:  87nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233577(3-(2-(1-(4-bromofuran-2-yl)propylamino)-3,4-dioxoc...)
Affinity DataIC50:  93nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233559(3-(2-(1-(5-((dimethylamino)methyl)furan-2-yl)propy...)
Affinity DataIC50:  94nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233553(2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylfuran-2-yl...)
Affinity DataIC50:  99nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233589(3-(2-(1-(4-chlorofuran-2-yl)propylamino)-3,4-dioxo...)
Affinity DataIC50:  100nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233561((R)-3-(3,4-dioxo-2-(1-(thiophen-3-yl)propylamino)c...)
Affinity DataIC50:  104nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233554((R)-3-(3,4-dioxo-2-(1-(pyridin-2-yl)propylamino)cy...)
Affinity DataIC50:  148nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233571(3-(3,4-dioxo-2-(1-(5-(2-(trifluoromethyl)phenyl)fu...)
Affinity DataIC50:  150nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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