Compile Data Set for Download or QSAR
maximum 50k data
Found 76 Enz. Inhib. hit(s) with all data for entry = 50025696
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251131(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-cycloh...)
Affinity DataIC50:  49.4nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251130(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-Ncyclohe...)
Affinity DataIC50:  62.8nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242549(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-cyclo...)
Affinity DataIC50:  66.5nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242548(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-cyclo...)
Affinity DataIC50:  72.8nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251131(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-cycloh...)
Affinity DataIC50:  82.3nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242557(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50:  89.2nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251130(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-Ncyclohe...)
Affinity DataIC50:  103nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242582(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50:  104nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50:  120nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242566(CHEMBL519584 | N-tert-Butyl-4-((2-chlorophenyl)(4-...)
Affinity DataIC50:  122nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251132(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-(cyclo...)
Affinity DataIC50:  127nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242548(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-cyclo...)
Affinity DataIC50:  128nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242601(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50:  141nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251132(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-(cyclo...)
Affinity DataIC50:  146nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242568(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-cycloheptylp...)
Affinity DataIC50:  151nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242537(4-((4-Chlorophenyl)(2,3-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50:  158nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242568(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-cycloheptylp...)
Affinity DataIC50:  163nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242600(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50:  163nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242600(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50:  186nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242556(4-((4-Chlorophenyl)(2,3-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50:  186nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242565(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-(cycl...)
Affinity DataIC50:  189nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242567(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-cyclohexylpi...)
Affinity DataIC50:  195nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242601(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50:  204nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251117(2-(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-pipe...)
Affinity DataIC50:  226nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242549(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-cyclo...)
Affinity DataIC50:  226nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251118(2-(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-pipe...)
Affinity DataIC50:  229nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251133(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-tert-b...)
Affinity DataIC50:  237nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242567(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-cyclohexylpi...)
Affinity DataIC50:  248nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242547(1-(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-...)
Affinity DataIC50:  257nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242558(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-(...)
Affinity DataIC50:  262nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242565(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-(cycl...)
Affinity DataIC50:  273nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251133(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-tert-b...)
Affinity DataIC50:  286nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242598(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-(cyclohexylm...)
Affinity DataIC50:  291nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242539(CHEMBL472299 | N-tert-Butyl-4-((4-chlorophenyl)(2,...)
Affinity DataIC50:  316nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242599(CHEMBL528325 | N-tert-Butyl-4-((4-chlorophenyl)(o-...)
Affinity DataIC50:  334nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242598(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-(cyclohexylm...)
Affinity DataIC50:  340nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242582(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50:  367nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242537(4-((4-Chlorophenyl)(2,3-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50:  424nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242556(4-((4-Chlorophenyl)(2,3-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50:  441nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242566(CHEMBL519584 | N-tert-Butyl-4-((2-chlorophenyl)(4-...)
Affinity DataIC50:  443nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251115(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50:  526nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242599(CHEMBL528325 | N-tert-Butyl-4-((4-chlorophenyl)(o-...)
Affinity DataIC50:  680nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242557(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50:  729nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242539(CHEMBL472299 | N-tert-Butyl-4-((4-chlorophenyl)(2,...)
Affinity DataIC50:  783nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251115(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50:  798nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242581(4-(Bis(4-chlorophenyl)methyl)-N-cyclohexylpiperazi...)
Affinity DataIC50:  914nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242558(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-(...)
Affinity DataIC50:  1.04E+3nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242584((4-(Bis(4-chlorophenyl)methyl)piperazin-1-yl)-(cyc...)
Affinity DataIC50:  1.07E+3nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242585(1-(4-(Bis(4-chlorophenyl)methyl)piperazin-1-yl)-he...)
Affinity DataIC50:  1.15E+3nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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