Compile Data Set for Download or QSAR
maximum 50k data
Found 244 Enz. Inhib. hit(s) with all data for entry = 50004135
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  650nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  975nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of recombinant Aurora AMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of recombinant VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  1.87E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  2.06E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  2.18E+3nMAssay Description:Inhibition of recombinant B-RAF-V600E mutantMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  2.21E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  2.22E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  2.48E+3nMAssay Description:Inhibition of recombinant CDK2/CycAMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  2.78E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  2.82E+3nMAssay Description:Inhibition of recombinant Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  2.87E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibition of recombinant IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.44E+3nMAssay Description:Inhibition of recombinant PDGFRbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50276157(Alternariol 5-O-Methyl Ether | CHEMBL483526)
Affinity DataIC50:  3.52E+3nMAssay Description:Inhibition of recombinant VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.56E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.67E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50276157(Alternariol 5-O-Methyl Ether | CHEMBL483526)
Affinity DataIC50:  3.67E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.71E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50576(2-(4,5-dihydroxy-2-methyl-phenyl)-6-hydroxy-4-meth...)
Affinity DataIC50:  3.78E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  3.81E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  3.81E+3nMAssay Description:Inhibition of recombinant EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  3.84E+3nMAssay Description:Inhibition of recombinant PDGFRbetaMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.87E+3nMAssay Description:Inhibition of recombinant FLT3 phosphorylation transfected in mouse embryonic fibroblastMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.87E+3nMAssay Description:Inhibition of recombinant IGF1R phosphorylation transfected in mouse embryonic fibroblastMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.87E+3nMAssay Description:Inhibition of recombinant VEGFR2 phosphorylation in human HUE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  3.87E+3nMAssay Description:Inhibition of recombinant Aurora B phosphorylation in human HT29 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  3.97E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50276157(Alternariol 5-O-Methyl Ether | CHEMBL483526)
Affinity DataIC50:  4.04E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50276157(Alternariol 5-O-Methyl Ether | CHEMBL483526)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of recombinant SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of recombinant INSRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50276157(Alternariol 5-O-Methyl Ether | CHEMBL483526)
Affinity DataIC50:  4.77E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of recombinant Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of recombinant IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  4.85E+3nMAssay Description:Inhibition of recombinant SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  4.85E+3nMAssay Description:Inhibition of recombinant TIE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479264(Alternariol 5-O-Sulfate | CHEMBL483525)
Affinity DataIC50:  5.02E+3nMAssay Description:Inhibition of recombinant VEGFR3More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479267(Alternariol | CHEBI:64983)
Affinity DataIC50:  5.03E+3nMAssay Description:Inhibition of recombinant VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50276157(Alternariol 5-O-Methyl Ether | CHEMBL483526)
Affinity DataIC50:  5.14E+3nMAssay Description:Inhibition of recombinant EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of recombinant Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479266(CHEMBL520144)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of recombinant B-RAF-V600E mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479263(Desmethylaltenusin)
Affinity DataIC50:  5.43E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50576(2-(4,5-dihydroxy-2-methyl-phenyl)-6-hydroxy-4-meth...)
Affinity DataIC50:  5.51E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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