Compile Data Set for Download or QSAR
maximum 50k data
Found 73 Enz. Inhib. hit(s) with all data for entry = 50038803
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186245((2S)-1-[(adamantan-1-yl)carbonyl]-N-{4-[4-(2-metho...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186236(Adamantane-1-carboxylic acid ((S)-1-{4-[4-(2-metho...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50267043(2-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2-az...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50026916(2-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2-a...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  6.05nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50206351((S)-N-(1-(4-(4-(3-chlorophenyl)piperazin-1-yl)buty...)
Affinity DataKi:  6.51nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186243(2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(4-(4-(2-me...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50267043(2-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2-az...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186255((S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphen...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186244((S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)but...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186253((S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphen...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50267016(CHEMBL514202 | N-[2-{4-(2-Methoxyphenyl)-piperazin...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50206351((S)-N-(1-(4-(4-(3-chlorophenyl)piperazin-1-yl)buty...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50001859((buspirone) 8-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186248(2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(3-(4-(2-me...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266905((S)-N-(1-(4-(4-(3-chlorophenyl)piperazin-1-yl)buty...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186243(2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(4-(4-(2-me...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186250(Adamantane-1-carboxylic acid ((S)-1-{3-[4-(2-metho...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186242((S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)but...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266905((S)-N-(1-(4-(4-(3-chlorophenyl)piperazin-1-yl)buty...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266983((S)-1-benzoyl-N-(4-(4-(3-chlorophenyl)piperazin-1-...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266845((S)-N-(1-(3-(4-(3-chlorophenyl)piperazin-1-yl)prop...)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266939((S)-N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-...)
Affinity DataKi:  111nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266983((S)-1-benzoyl-N-(4-(4-(3-chlorophenyl)piperazin-1-...)
Affinity DataKi:  128nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50267042(CHEMBL477945 | N-[2-{4-(3-Chlorophenyl)-piperazin-...)
Affinity DataKi:  137nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266939((S)-N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-...)
Affinity DataKi:  163nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186236(Adamantane-1-carboxylic acid ((S)-1-{4-[4-(2-metho...)
Affinity DataKi:  173nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186244((S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)but...)
Affinity DataKi:  183nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50267042(CHEMBL477945 | N-[2-{4-(3-Chlorophenyl)-piperazin-...)
Affinity DataKi:  227nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186241((S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)pro...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50026916(2-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2-a...)
Affinity DataKi:  254nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266818((S)-1-(Adamantane-1-carbonyl)-pyrrolidine-2-carbox...)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266844((S)-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-...)
Affinity DataKi:  357nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266845((S)-N-(1-(3-(4-(3-chlorophenyl)piperazin-1-yl)prop...)
Affinity DataKi:  360nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266872((S)-1-benzoyl-N-(3-(4-(2-methoxyphenyl)piperazin-1...)
Affinity DataKi:  390nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186237((S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)pro...)
Affinity DataKi:  480nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266718(2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(2-(4-(2-me...)
Affinity DataKi:  497nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186245((2S)-1-[(adamantan-1-yl)carbonyl]-N-{4-[4-(2-metho...)
Affinity DataKi:  503nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266719(Adamantane-1-carboxylic acid ((S)-1-{2-[4-(2-metho...)
Affinity DataKi:  579nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266904((S)-1-acetyl-N-(3-(4-(2-methoxyphenyl)piperazin-1-...)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266871((S)-N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50267016(CHEMBL514202 | N-[2-{4-(2-Methoxyphenyl)-piperazin...)
Affinity DataKi:  868nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50186253((S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphen...)
Affinity DataKi:  990nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266721((S)-1-(cyclohexanecarbonyl)-N-(2-(4-(2-methoxyphen...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266815((S)-1-benzoyl-N-(2-(4-(3-chlorophenyl)piperazin-1-...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50267228((S)-N-(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethy...)
Affinity DataKi:  1.41E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266741((S)-1-benzoyl-N-(2-(4-(2-methoxyphenyl)piperazin-1...)
Affinity DataKi:  1.51E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266871((S)-N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)...)
Affinity DataKi:  1.73E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat hippocampal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50267229((S)-N-(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethy...)
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50266818((S)-1-(Adamantane-1-carbonyl)-pyrrolidine-2-carbox...)
Affinity DataKi:  1.92E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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