Compile Data Set for Download or QSAR
maximum 50k data
Found 88 Enz. Inhib. hit(s) with all data for entry = 50026627
LigandPNGBDBM50262463((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-7,7-di...)
Affinity DataIC50:  18nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262463((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-7,7-di...)
Affinity DataIC50:  31nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262460((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  35nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262460((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  49nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262460((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  51nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262463((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-7,7-di...)
Affinity DataIC50:  59nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262462((S)-2-(3-(benzo[b]thiophen-3-ylmethyl)morpholino)-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262461(2-(3-((1H-pyrrolo[2,3-b]pyridin-3-yl)methyl)morpho...)
Affinity DataIC50:  63nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262461(2-(3-((1H-pyrrolo[2,3-b]pyridin-3-yl)methyl)morpho...)
Affinity DataIC50:  74nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262461(2-(3-((1H-pyrrolo[2,3-b]pyridin-3-yl)methyl)morpho...)
Affinity DataIC50:  107nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262462((S)-2-(3-(benzo[b]thiophen-3-ylmethyl)morpholino)-...)
Affinity DataIC50:  125nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262408(5,5-dimethyl-2-(3-(naphthalen-1-ylmethyl)morpholin...)
Affinity DataIC50:  126nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262463((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-7,7-di...)
Affinity DataIC50:  199nMAssay Description:Inhibition of PI3K-mediated AKT Ser473 phosphorylation in PTEN negative human MCF7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262462((S)-2-(3-(benzo[b]thiophen-3-ylmethyl)morpholino)-...)
Affinity DataIC50:  223nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262408(5,5-dimethyl-2-(3-(naphthalen-1-ylmethyl)morpholin...)
Affinity DataIC50:  229nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262408(5,5-dimethyl-2-(3-(naphthalen-1-ylmethyl)morpholin...)
Affinity DataIC50:  386nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262461(2-(3-((1H-pyrrolo[2,3-b]pyridin-3-yl)methyl)morpho...)
Affinity DataIC50:  481nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261834(2-morpholin-4-yl-5,6-dihydro-4H-benzothiazol-7-one...)
Affinity DataIC50:  693nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261834(2-morpholin-4-yl-5,6-dihydro-4H-benzothiazol-7-one...)
Affinity DataIC50:  701nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262407((S)-2-(3-benzylmorpholino)-5,5-dimethyl-5,6-dihydr...)
Affinity DataIC50:  833nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261834(2-morpholin-4-yl-5,6-dihydro-4H-benzothiazol-7-one...)
Affinity DataIC50:  975nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262463((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-7,7-di...)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262460((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262354(2-(morpholin-4-yl)-6,7-dihydro-4H-spiro[1,3-benzot...)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262353(2-(morpholin-4-yl)-6,7-dihydro-4H-spiro[1,3-benzot...)
Affinity DataIC50:  1.28E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262409(5,5-dimethyl-2-(3-(naphthalen-2-ylmethyl)morpholin...)
Affinity DataIC50:  1.39E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262463((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-7,7-di...)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of PI3K-mediated AKT Ser473 phosphorylation in PTEN negative human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262353(2-(morpholin-4-yl)-6,7-dihydro-4H-spiro[1,3-benzot...)
Affinity DataIC50:  1.48E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262460((S)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of PI3K-mediated AKT Ser473 phosphorylation in PTEN negative human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262354(2-(morpholin-4-yl)-6,7-dihydro-4H-spiro[1,3-benzot...)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262409(5,5-dimethyl-2-(3-(naphthalen-2-ylmethyl)morpholin...)
Affinity DataIC50:  1.67E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262354(2-(morpholin-4-yl)-6,7-dihydro-4H-spiro[1,3-benzot...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262407((S)-2-(3-benzylmorpholino)-5,5-dimethyl-5,6-dihydr...)
Affinity DataIC50:  2.08E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262407((S)-2-(3-benzylmorpholino)-5,5-dimethyl-5,6-dihydr...)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262353(2-(morpholin-4-yl)-6,7-dihydro-4H-spiro[1,3-benzot...)
Affinity DataIC50:  2.43E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262296(CHEMBL466956 | rac-5-methyl-2-morpholino-5,6-dihyd...)
Affinity DataIC50:  2.49E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262410((R)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  2.53E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262462((S)-2-(3-(benzo[b]thiophen-3-ylmethyl)morpholino)-...)
Affinity DataIC50:  2.55E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262410((R)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  2.56E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261834(2-morpholin-4-yl-5,6-dihydro-4H-benzothiazol-7-one...)
Affinity DataIC50:  2.94E+3nMAssay Description:Inhibition of PI3K-mediated AKT Ser473 phosphorylation in PTEN negative human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50261834(2-morpholin-4-yl-5,6-dihydro-4H-benzothiazol-7-one...)
Affinity DataIC50:  3.45E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
LigandPNGBDBM50262409(5,5-dimethyl-2-(3-(naphthalen-2-ylmethyl)morpholin...)
Affinity DataIC50:  3.49E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262410((R)-2-(3-((1H-indol-3-yl)methyl)morpholino)-5,5-di...)
Affinity DataIC50:  3.51E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262299(2-morpholino-5,6-dihydrobenzo[d]thiazol-7(4H)-one ...)
Affinity DataIC50:  3.58E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262299(2-morpholino-5,6-dihydrobenzo[d]thiazol-7(4H)-one ...)
Affinity DataIC50:  3.89E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262357(5,5-dimethyl-2-(pyridin-4-yl)-5,6-dihydrobenzo[d]t...)
Affinity DataIC50:  4.16E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262296(CHEMBL466956 | rac-5-methyl-2-morpholino-5,6-dihyd...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262296(CHEMBL466956 | rac-5-methyl-2-morpholino-5,6-dihyd...)
Affinity DataIC50:  5.97E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262354(2-(morpholin-4-yl)-6,7-dihydro-4H-spiro[1,3-benzot...)
Affinity DataIC50:  6.26E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50262408(5,5-dimethyl-2-(3-(naphthalen-1-ylmethyl)morpholin...)
Affinity DataIC50:  6.94E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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