Compile Data Set for Download or QSAR
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Found 15 Enz. Inhib. hit(s) with all data for entry = 50000772
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataKi:  3.60nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataKi:  16nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataKi:  50nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009674(4-Amino-N-[2-(4-amino-butyrylamino)-ethyl]-N-[2-((...)
Affinity DataKi:  3.73E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009677(4-Amino-N-[3-(4-amino-butyrylamino)-propyl]-N-{3-[...)
Affinity DataKi:  5.51E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009674(4-Amino-N-[2-(4-amino-butyrylamino)-ethyl]-N-[2-((...)
Affinity DataKi:  6.76E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009677(4-Amino-N-[3-(4-amino-butyrylamino)-propyl]-N-{3-[...)
Affinity DataKi:  7.30E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009677(4-Amino-N-[3-(4-amino-butyrylamino)-propyl]-N-{3-[...)
Affinity DataKi:  8.43E+3nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009678(4-Amino-N-[2-(4-amino-butyrylamino)-ethyl]-N-{2-[2...)
Affinity DataKi:  8.75E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009674(4-Amino-N-[2-(4-amino-butyrylamino)-ethyl]-N-[2-((...)
Affinity DataKi: >1.00E+4nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009676(4-Amino-N-{2-[2-(2-{2-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKi:  1.01E+4nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009678(4-Amino-N-[2-(4-amino-butyrylamino)-ethyl]-N-{2-[2...)
Affinity DataKi:  1.44E+4nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009676(4-Amino-N-{2-[2-(2-{2-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKi:  1.65E+4nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009678(4-Amino-N-[2-(4-amino-butyrylamino)-ethyl]-N-{2-[2...)
Affinity DataKi:  2.27E+4nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Case Western Reserve University

Curated by ChEMBL
LigandPNGBDBM50009676(4-Amino-N-{2-[2-(2-{2-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKi:  3.67E+4nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed