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Found 24 Enz. Inhib. hit(s) with all data for entry = 50027601
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279520(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-p...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279541(2-(4-(4-(1H-indol-3-yl)piperidin-1-yl)butyl)-4-(2-...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279541(2-(4-(4-(1H-indol-3-yl)piperidin-1-yl)butyl)-4-(2-...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279520(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-p...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279540(4-(4-Fluoro-phenyl)-2-{4-[4-(1H-indol-3-yl)-piperi...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279561(2-(4-(4-(1H-indol-3-yl)piperidin-1-yl)butyl)-4-phe...)
Affinity DataKi:  10.9nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279586(4-(2-fluorophenyl)-2-(4-(4-(5-methoxy-1H-indol-3-y...)
Affinity DataKi:  16.7nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279585(4-(4-fluorophenyl)-2-(4-(4-(5-methoxy-1H-indol-3-y...)
Affinity DataKi:  34.6nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279539(4-(4-Chloro-phenyl)-2-{4-[4-(1H-indol-3-yl)-piperi...)
Affinity DataKi:  37.1nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279540(4-(4-Fluoro-phenyl)-2-{4-[4-(1H-indol-3-yl)-piperi...)
Affinity DataKi:  37.6nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279564(4-(4-chlorophenyl)-2-(4-(4-(5-methoxy-1H-indol-3-y...)
Affinity DataKi:  41.1nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279519(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-(...)
Affinity DataKi:  42.1nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279587(2-(4-(4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl)bu...)
Affinity DataKi:  52.3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279585(4-(4-fluorophenyl)-2-(4-(4-(5-methoxy-1H-indol-3-y...)
Affinity DataKi:  54.6nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279561(2-(4-(4-(1H-indol-3-yl)piperidin-1-yl)butyl)-4-phe...)
Affinity DataKi:  58.1nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279563(2-(4-(4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl)bu...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279586(4-(2-fluorophenyl)-2-(4-(4-(5-methoxy-1H-indol-3-y...)
Affinity DataKi:  59.3nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279562(2-(4-(4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl)bu...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279587(2-(4-(4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl)bu...)
Affinity DataKi:  129nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279562(2-(4-(4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl)bu...)
Affinity DataKi:  129nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279519(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-(...)
Affinity DataKi:  145nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279563(2-(4-(4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl)bu...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279564(4-(4-chlorophenyl)-2-(4-(4-(5-methoxy-1H-indol-3-y...)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279539(4-(4-Chloro-phenyl)-2-{4-[4-(1H-indol-3-yl)-piperi...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed