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Found 9 Enz. Inhib. hit(s) with all data for entry = 50038717
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50377962(CAMBOGIN)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of HAT p300 catalytic domain by equilibrium dialysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50241990(CHEMBL502489 | Camboginol | Garcinol | Garcinol, 1)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of HAT p300 catalytic domain by equilibrium dialysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50265449((1R,3S,9S,11R)-7-(3-Hydroxy-4-methoxy-benzoyl)-4,4...)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of HAT p300 catalytic domain by equilibrium dialysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50241990(CHEMBL502489 | Camboginol | Garcinol | Garcinol, 1)
Affinity DataKd:  6.60E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50377962(CAMBOGIN)
Affinity DataKd:  5.90E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50377962(CAMBOGIN)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by fluorometric titrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50265449((1R,3S,9S,11R)-7-(3-Hydroxy-4-methoxy-benzoyl)-4,4...)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by fluorometric titrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50241990(CHEMBL502489 | Camboginol | Garcinol | Garcinol, 1)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by fluorometric titrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50265449((1R,3S,9S,11R)-7-(3-Hydroxy-4-methoxy-benzoyl)-4,4...)
Affinity DataKd:  9.10E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed