Compile Data Set for Download or QSAR
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Found 42 Enz. Inhib. hit(s) with all data for entry = 50041691
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413253(CHEMBL470587)
Affinity DataEC50:  100nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413273(CHEMBL471421)
Affinity DataEC50:  126nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413255(CHEMBL513760)
Affinity DataEC50:  19.9nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413256(CHEMBL472476)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413257(CHEMBL469322)
Affinity DataEC50:  251nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413258(CHEMBL469281)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413259(CHEMBL469323)
Affinity DataEC50:  31.6nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413260(CHEMBL198794)
Affinity DataEC50:  15.8nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413261(AC-55649 | CHEMBL425027)
Affinity DataEC50:  126nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)
Affinity DataEC50:  19.9nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50:  6.31nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50:  25.1nMAssay Description:Activity at RARbeta1 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)
Affinity DataEC50:  50.1nMAssay Description:Activity at RARbeta1 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413253(CHEMBL470587)
Affinity DataEC50:  1.00E+3nMAssay Description:Activity at RARbeta1 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413260(CHEMBL198794)
Affinity DataEC50:  316nMAssay Description:Activity at RARbeta1 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413261(AC-55649 | CHEMBL425027)
Affinity DataEC50:  2.00E+3nMAssay Description:Activity at RARbeta1 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413262(CHEMBL472032)
Affinity DataEC50:  100nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413263(CHEMBL472213)
Affinity DataEC50:  100nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413264(CHEMBL472236)
Affinity DataEC50:  631nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413265(CHEMBL524687)
Affinity DataEC50:  39.8nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413266(CHEMBL471197)
Affinity DataEC50:  126nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413267(CHEMBL371684)
Affinity DataEC50:  25.1nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413268(CHEMBL471423)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413269(CHEMBL471422)
Affinity DataEC50:  79.4nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413270(CHEMBL512879)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413271(CHEMBL472238)
Affinity DataEC50:  39.8nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413272(AC-261066 | CHEMBL198997)
Affinity DataEC50:  7.94nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413261(AC-55649 | CHEMBL425027)
Affinity DataEC50:  2.51E+3nMAssay Description:Activity at RARalpha expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413265(CHEMBL524687)
Affinity DataEC50:  2.00E+3nMAssay Description:Activity at RARalpha expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413255(CHEMBL513760)
Affinity DataEC50:  1.58E+3nMAssay Description:Activity at RARalpha expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)
Affinity DataEC50:  79.4nMAssay Description:Activity at RARalpha expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413272(AC-261066 | CHEMBL198997)
Affinity DataEC50:  631nMAssay Description:Activity at RARalpha expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413265(CHEMBL524687)
Affinity DataEC50:  398nMAssay Description:Activity at RARbeta1 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413272(AC-261066 | CHEMBL198997)
Affinity DataEC50:  398nMAssay Description:Activity at RARbeta1 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413269(CHEMBL471422)
Affinity DataEC50:  1.26E+3nMAssay Description:Activity at RARbeta1 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)
Affinity DataEC50:  25.1nMAssay Description:Activity at RARgamma expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413272(AC-261066 | CHEMBL198997)
Affinity DataEC50:  501nMAssay Description:Activity at RARgamma expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413271(CHEMBL472238)
Affinity DataEC50:  631nMAssay Description:Activity at RARgamma expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413265(CHEMBL524687)
Affinity DataEC50:  158nMAssay Description:Activity at RARgamma expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50:  50.1nMAssay Description:Activity at RARgamma expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50:  6.31nMAssay Description:Activity at RARalpha expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413254(CHEMBL470588)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed