TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Antagonist activity at MCH1R (unknown origin)More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataKi: 3.16nMAssay Description:Antagonist activity at MCH1R (unknown origin)More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Antagonist activity at MCH1R (unknown origin)More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataKi: 77nMAssay Description:Antagonist activity at MCH1R (unknown origin)More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataKi: 164nMAssay Description:Antagonist activity at MCH1R (unknown origin)More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Antagonist activity at MCH1R (unknown origin)More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Antagonist activity at MCH1R (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at MCH1R (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Antagonist activity at MCH1R (unknown origin)More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Antagonist activity at MCH1R (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataIC50: 1.17E+3nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Antagonist activity at MCH1R (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Johnson & Johnson Pharmaceutical R&D
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair