Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50028519
TargetVitamin D3 receptor(Homo sapiens (Human))
Bioxell

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  10nMAssay Description:Activation of VDR in human THP1 cells assessed as increase in 25-hydroxyvitamin D-24-hydroxylase mRNA expression by RT-PCRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetVitamin D3 receptor(Homo sapiens (Human))
Bioxell

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  10nMAssay Description:Activation of VDR in human THP1 cells assessed as increase in cathelicidin antimicrobial peptide mRNA expression by RT-PCRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetVitamin D3 receptor(Homo sapiens (Human))
Bioxell

Curated by ChEMBL
LigandPNGBDBM50293274(1alpha,25(OH)2-24-oxo-16-ene-20-cyclopropyl-vitami...)
Affinity DataEC50:  0.690nMAssay Description:Activation of VDR in human THP1 cells assessed as increase in cathelicidin antimicrobial peptide mRNA expression by RT-PCRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Bioxell

Curated by ChEMBL
LigandPNGBDBM50257431(1,25-dihydroxy-16-ene-20-cyclopropyl-vitamin D3 | ...)
Affinity DataEC50:  0.680nMAssay Description:Activation of VDR in human THP1 cells assessed as increase in cathelicidin antimicrobial peptide mRNA expression by RT-PCRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Bioxell

Curated by ChEMBL
LigandPNGBDBM50293274(1alpha,25(OH)2-24-oxo-16-ene-20-cyclopropyl-vitami...)
Affinity DataEC50:  0.690nMAssay Description:Activation of VDR in human THP1 cells assessed as increase in 25-hydroxyvitamin D-24-hydroxylase mRNA expression by RT-PCRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Bioxell

Curated by ChEMBL
LigandPNGBDBM50257431(1,25-dihydroxy-16-ene-20-cyclopropyl-vitamin D3 | ...)
Affinity DataEC50:  0.680nMAssay Description:Activation of VDR in human THP1 cells assessed as increase in 25-hydroxyvitamin D-24-hydroxylase mRNA expression by RT-PCRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed