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Found 58 Enz. Inhib. hit(s) with all data for entry = 50041734
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414353(CHEMBL563425)
Affinity DataKi:  2.88nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414355(CHEMBL560624)
Affinity DataKi:  3.02nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414354(CHEMBL551904)
Affinity DataKi:  3.02nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414358(CHEMBL557694)
Affinity DataKi:  9.12nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414351(CHEMBL561364)
Affinity DataKi:  11.8nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414362(CHEMBL556389)
Affinity DataKi:  15.5nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414360(CHEMBL562427)
Affinity DataKi:  15.5nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414357(CHEMBL560905)
Affinity DataKi:  20.9nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414354(CHEMBL551904)
Affinity DataKi:  20.9nMAssay Description:Binding affinity to rat cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414352(CHEMBL552304)
Affinity DataKi:  33.9nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414355(CHEMBL560624)
Affinity DataKi:  36.3nMAssay Description:Binding affinity to rat cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414356(CHEMBL565192)
Affinity DataKi:  49.0nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414354(CHEMBL551904)
Affinity DataKi:  56.2nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414368(CHEMBL563889)
Affinity DataKi:  70.8nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414363(CHEMBL560623)
Affinity DataKi:  77.6nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414367(CHEMBL560967)
Affinity DataKi:  85.1nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414355(CHEMBL560624)
Affinity DataKi:  87.1nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414361(CHEMBL550638)
Affinity DataKi:  93.3nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414357(CHEMBL560905)
Affinity DataKi:  95.5nMAssay Description:Binding affinity to rat cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414352(CHEMBL552304)
Affinity DataKi:  95.5nMAssay Description:Binding affinity to human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414363(CHEMBL560623)
Affinity DataKi:  95.5nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414353(CHEMBL563425)
Affinity DataKi:  97.7nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414356(CHEMBL565192)
Affinity DataKi:  100nMAssay Description:Binding affinity to rat cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414353(CHEMBL563425)
Affinity DataKi:  100nMAssay Description:Binding affinity to rat cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414358(CHEMBL557694)
Affinity DataKi:  112nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414369(CHEMBL564680)
Affinity DataKi:  126nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414370(CHEMBL551761)
Affinity DataKi:  138nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414351(CHEMBL561364)
Affinity DataKi:  148nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414365(CHEMBL561168)
Affinity DataKi:  148nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414352(CHEMBL552304)
Affinity DataKi:  162nMAssay Description:Binding affinity to rat cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414362(CHEMBL556389)
Affinity DataKi:  170nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414359(CHEMBL563259)
Affinity DataKi:  174nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414360(CHEMBL562427)
Affinity DataKi:  174nMAssay Description:Binding affinity to rat cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414361(CHEMBL550638)
Affinity DataKi:  204nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414367(CHEMBL560967)
Affinity DataKi:  209nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414359(CHEMBL563259)
Affinity DataKi:  209nMAssay Description:Binding affinity to human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414357(CHEMBL560905)
Affinity DataKi:  214nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414369(CHEMBL564680)
Affinity DataKi:  219nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414356(CHEMBL565192)
Affinity DataKi:  229nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414366(CHEMBL561167)
Affinity DataKi:  324nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414366(CHEMBL561167)
Affinity DataKi:  339nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414358(CHEMBL557694)
Affinity DataKi:  398nMAssay Description:Binding affinity to human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414365(CHEMBL561168)
Affinity DataKi:  398nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414360(CHEMBL562427)
Affinity DataKi:  417nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414364(CHEMBL556264)
Affinity DataKi:  490nMAssay Description:Binding affinity to human adenosine A2b receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414370(CHEMBL551761)
Affinity DataKi:  490nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414368(CHEMBL563889)
Affinity DataKi:  525nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414358(CHEMBL557694)
Affinity DataKi:  676nMAssay Description:Binding affinity to rat cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414351(CHEMBL561364)
Affinity DataKi:  708nMAssay Description:Binding affinity to human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50414352(CHEMBL552304)
Affinity DataKi:  759nMAssay Description:Binding affinity to human adenosine A2a receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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