Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50041745
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | CHEM...)
Affinity DataIC50:  1.29nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50:  45.7nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414658(CHEMBL559048)
Affinity DataIC50:  58.9nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414645(CYASTERONE)
Affinity DataIC50:  61.7nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414646(INOKOSTERONE)
Affinity DataIC50:  91.2nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50226672(CHEMBL255034 | makisterone A)
Affinity DataIC50:  112nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414659(CHEMBL564892)
Affinity DataIC50:  324nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414652(CHEMBL559941)
Affinity DataIC50:  794nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414651(ECDYSONE)
Affinity DataIC50:  2.57E+3nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414655(CHEMBL560796)
Affinity DataIC50:  9.55E+3nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414657(CHEMBL562711)
Affinity DataIC50:  1.45E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414660(CHEMBL564474)
Affinity DataIC50:  3.89E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414649(CHEMBL561275)
Affinity DataIC50:  4.17E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414647(CHEMBL560194)
Affinity DataIC50:  4.17E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414653(CHEMBL558256)
Affinity DataIC50:  8.91E+4nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414654(CHEMBL560139)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414650(CHEMBL550600)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414648(CHEMBL559545)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414656(CHEMBL558652)
Affinity DataIC50: >2.45E+5nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed