Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 50030942
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304315(CHEMBL593465 | trans-3-Oxo-N-(2-phenyl-2H-1,2,3-tr...)
Affinity DataIC50:  0.890nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304301(CHEMBL595790 | trans-N-[1-(3-Fluorophenyl)-1H-pyra...)
Affinity DataIC50:  0.920nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304313(CHEMBL607037 | trans-3-Oxo-N-(2-phenyl-1,3-thiazol...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304298(CHEMBL595120 | trans-3-Oxo-N-(1-phenyl-1H-pyrazol-...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304300(CHEMBL595573 | trans-N-[1-(2-fluorophenyl)-3-pyraz...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304303(CHEMBL593934 | trans-3-Oxo-N-(5-phenylpyrazin-2-yl...)
Affinity DataIC50:  1.5nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Rat 6B)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304297(CHEMBL594163 | trans-3-Oxo-N-(1-phenyl-1H-pyrazol-...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301656(CHEMBL567527 | trans-1'-oxo-N-(5-phenylpyrimidin-2...)
Affinity DataIC50:  1.80nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304316(CHEMBL594164 | trans-N-[1-(4-Fluorophenyl)-1H-pyra...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301651(CHEMBL568370 | trans-3'-oxo-N-(5-phenylpyrimidin-2...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304310(CHEMBL596264 | trans-3-Oxo-N-(5-phenylisoxazol-3-y...)
Affinity DataIC50:  2.10nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304312(CHEMBL604480 | trans-3-Oxo-N-(5-phenylpyridin-2-yl...)
Affinity DataIC50:  2.10nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Rat 6B)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304301(CHEMBL595790 | trans-N-[1-(3-Fluorophenyl)-1H-pyra...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Rat 6B)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304300(CHEMBL595573 | trans-N-[1-(2-fluorophenyl)-3-pyraz...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301644(CHEMBL568144 | trans-3-Oxo-N-(5-phenylpyrimidin-2-...)
Affinity DataIC50:  2.10nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304309(CHEMBL607144 | trans-3-Oxo-N-(5-phenylpyrazin-2-yl...)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Rat 6B)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304299(CHEMBL595560 | trans-3-Oxo-N-(1-phenyl-1H-pyrazol-...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304314(CHEMBL596025 | trans-3-Oxo-N-(1-phenyl-1H-pyrazol-...)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304299(CHEMBL595560 | trans-3-Oxo-N-(1-phenyl-1H-pyrazol-...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304318(CHEMBL594888 | trans-3-Oxo-N-(5-phenylisoxazol-3-y...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304307(CHEMBL595121 | trans-3-Oxo-N-(5-phenylpyrazin-2-yl...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Rat 6B)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304302(3'-oxo-N-(5-phenylpyrazin-2-yl)-3'H-spiro[cyclohex...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304311(CHEMBL606631 | trans-3-Oxo-N-(3-phenyl-1H-pyrazol-...)
Affinity DataIC50:  2.70nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304305(CHEMBL607192 | trans-3-Oxo-N-(5-phenylisoxazol-3-y...)
Affinity DataIC50:  2.80nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304308(CHEMBL596266 | trans-3-Oxo-N-(3-phenyl-1H-pyrazol-...)
Affinity DataIC50:  2.90nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301641(CHEMBL585851 | trans-3-Oxo-N-(5-phenylpyrimidin-2-...)
Affinity DataIC50:  2.90nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304317(CHEMBL593466 | trans-3-Oxo-N-(5-phenylpyrazin-2-yl...)
Affinity DataIC50:  3.90nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304304(CHEMBL596031 | trans-3-Oxo-N-(5-phenylpyrazin-2-yl...)
Affinity DataIC50:  4.20nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304297(CHEMBL594163 | trans-3-Oxo-N-(1-phenyl-1H-pyrazol-...)
Affinity DataIC50:  4.40nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Rat 6B)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304298(CHEMBL595120 | trans-3-Oxo-N-(1-phenyl-1H-pyrazol-...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of rat Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304306(CHEMBL607088 | trans-3-Oxo-N-(3-phenyl-1H-pyrazol-...)
Affinity DataIC50:  5.40nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50304319(CHEMBL593935 | trans-3-Oxo-N-(3-phenyl-1H-pyrazol-...)
Affinity DataIC50:  26nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed