Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 3444
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Universite De Lyon

LigandPNGBDBM34110(glucopyranosylidene-spiro-isoxazoline, 4e)
Affinity DataKi:  630nM ΔG°:  -36.0kJ/molepH: 6.8 T: 2°CAssay Description:Phosphorylase activity was measured in the direction of glycogen synthesis by the release of orthophosphate from Glc-1-P. The enzyme was assayed in g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Universite De Lyon

LigandPNGBDBM34106(glucopyranosylidene-spiro-isoxazoline, 4a)
Affinity DataKi:  6.60E+3nM ΔG°:  -30.1kJ/molepH: 6.8 T: 2°CAssay Description:Phosphorylase activity was measured in the direction of glycogen synthesis by the release of orthophosphate from Glc-1-P. The enzyme was assayed in g...More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Universite De Lyon

LigandPNGBDBM34107(glucopyranosylidene-spiro-isoxazoline, 4b)
Affinity DataKi:  7.90E+3nM ΔG°:  -29.6kJ/molepH: 6.8 T: 2°CAssay Description:Phosphorylase activity was measured in the direction of glycogen synthesis by the release of orthophosphate from Glc-1-P. The enzyme was assayed in g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Universite De Lyon

LigandPNGBDBM34108(glucopyranosylidene-spiro-isoxazoline, 4c)
Affinity DataKi:  1.96E+4nM ΔG°:  -27.3kJ/molepH: 6.8 T: 2°CAssay Description:Phosphorylase activity was measured in the direction of glycogen synthesis by the release of orthophosphate from Glc-1-P. The enzyme was assayed in g...More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Universite De Lyon

LigandPNGBDBM34109(glucopyranosylidene-spiro-isoxazoline, 4d)
Affinity DataKi:  9.25E+4nM ΔG°:  -23.4kJ/molepH: 6.8 T: 2°CAssay Description:Phosphorylase activity was measured in the direction of glycogen synthesis by the release of orthophosphate from Glc-1-P. The enzyme was assayed in g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed