Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50048849
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataKi:  4nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228839(CHEMBL415414)
Affinity DataKi:  170nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50216682(1-(5-Isoquinolinesulfonyl)-2-methylpiperazine | 1-...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50216682(1-(5-Isoquinolinesulfonyl)-2-methylpiperazine | 1-...)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of ATP from protein kinase C (PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataIC50:  3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228839(CHEMBL415414)
Affinity DataIC50:  300nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228847(CHEMBL407100)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228838(CHEMBL428973)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228846(CHEMBL265876)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228841(CHEMBL351282)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50011236(CHEMBL344314 | Isoquinoline-5-sulfonic acid (2-ami...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50216682(1-(5-Isoquinolinesulfonyl)-2-methylpiperazine | 1-...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM15203(5-(piperazine-1-sulfonyl)isoquinoline | CHEMBL7577...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM15203(5-(piperazine-1-sulfonyl)isoquinoline | CHEMBL7577...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of protein kinase C (PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228844(CHEMBL263188)
Affinity DataIC50: >7.50E+4nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228842(CHEMBL437640)
Affinity DataIC50: >7.50E+4nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228845(CHEMBL410778)
Affinity DataIC50: >7.50E+4nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed