Compile Data Set for Download or QSAR
maximum 50k data
Found 66 Enz. Inhib. hit(s) with all data for entry = 50039105
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313446(CHEMBL1096003 | N-(((2R,4aS,5R,10bS)-9-chloro-7-fl...)
Affinity DataIC50:  2nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313441(3-(dimethylamino)-N-(((2R,4aS,5R,10bS)-9-isopropyl...)
Affinity DataIC50:  2nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313442(1-((2R,4aS,5R,10bS)-9-bromo-7-fluoro-5-phenyl-3,4,...)
Affinity DataIC50:  3nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313435(4-((2R,4aS,5R,10bS)-2-((methylamino)methyl)-9-(tri...)
Affinity DataIC50:  4nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313437(1-((2R,4aS,5R,10bS)-9-tert-butyl-5-phenyl-3,4,4a,5...)
Affinity DataIC50:  4nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313430(2-(methylamino)-N-(((2R,4aS,5R,10bS)-5-phenyl-9-(t...)
Affinity DataIC50:  4nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313444(CHEMBL1085692 | N-(((2R,4aS,5R,10bS)-9-bromo-7-flu...)
Affinity DataIC50:  5nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313439(1-((2R,4aS,5R,10bS)-9-tert-butyl-5-(thiophen-2-yl)...)
Affinity DataIC50:  5nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313434((2R,4aS,5R,10bS)-2-((1H-1,2,4-triazol-1-yl)methyl)...)
Affinity DataIC50:  6nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313443(CHEMBL1082249 | N-(2-(((2R,4aS,5R,10bS)-9-bromo-7-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313431(3-amino-N-methyl-N-(((2R,4aS,5R,10bS)-5-phenyl-9-(...)
Affinity DataIC50:  7nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313445(2-(((2R,4aS,5R,10bS)-9-chloro-7-fluoro-5-phenyl-3,...)
Affinity DataIC50:  7nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313428(1-(2-(dimethylamino)ethyl)-3-(((2R,4aS,5R,10bS)-5-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313440(1-((2R,4aS,5R,10bS)-9-cyclopropyl-5-phenyl-3,4,4a,...)
Affinity DataIC50:  11nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313427(1-(3-hydroxypropyl)-3-(((2R,4aS,5R,10bS)-5-phenyl-...)
Affinity DataIC50:  11nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313429(2-(dimethylamino)ethyl((2R,4aS,5R,10bS)-5-phenyl-9...)
Affinity DataIC50:  14nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313409(4-((4aS,5R,10bS)-9-tert-butyl-3,4,4a,5,6,10b-hexah...)
Affinity DataIC50:  17nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313432(CHEMBL1093087 | N1-phenyl-N1-(((2R,4aS,5R,10bS)-5-...)
Affinity DataIC50:  19nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313438(2-((((2R,4aS,5R,10bS)-9-tert-butyl-5-phenyl-3,4,4a...)
Affinity DataIC50:  19nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313426(((2R,4aS,5R,10bS)-5-phenyl-9-(trifluoromethyl)-3,4...)
Affinity DataIC50:  20nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313418((4aS,5R,10bS)-9-tert-butyl-5-(thiophen-2-yl)-3,4,4...)
Affinity DataIC50:  25nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313407(4-((4aS,5R,10bS)-9-tert-butyl-3,4,4a,5,6,10b-hexah...)
Affinity DataIC50:  34nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313406(3-((4aS,5R,10bS)-9-tert-butyl-3,4,4a,5,6,10b-hexah...)
Affinity DataIC50:  40nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313436(1-((2R,4aS,5R,10bS)-5-(4-fluorophenyl)-9-(trifluor...)
Affinity DataIC50:  58nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313433(CHEMBL1084431 | N-(2-aminoethyl)-4-methyl-N-(((2R,...)
Affinity DataIC50:  65nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313401((4aS,5R,10bS)-7-fluoro-5-phenyl-9-(trifluoromethyl...)
Affinity DataIC50:  90nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313408(4-((4aS,5R,10bS)-9-tert-butyl-3,4,4a,5,6,10b-hexah...)
Affinity DataIC50:  95nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313391((4aS,5R,10bS)-5-phenyl-9-(trifluoromethyl)-3,4,4a,...)
Affinity DataIC50:  110nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313419((4aS,5R,10bS)-9-tert-butyl-5-(thiophen-3-yl)-3,4,4...)
Affinity DataIC50:  120nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313387((4aS,5R,10bS)-9-ethyl-5-phenyl-3,4,4a,5,6,10b-hexa...)
Affinity DataIC50:  130nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313389((4aS,5R,10bS)-9-isopropyl-5-phenyl-3,4,4a,5,6,10b-...)
Affinity DataIC50:  130nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313414((4aS,5R,10bS)-9-tert-butyl-5-(2-fluorophenyl)-3,4,...)
Affinity DataIC50:  170nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313415((4aS,5R,10bS)-9-tert-butyl-5-(4-fluorophenyl)-3,4,...)
Affinity DataIC50:  270nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313390((4aS,5R,10bS)-9-tert-butyl-5-phenyl-3,4,4a,5,6,10b...)
Affinity DataIC50:  300nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313390((4aS,5R,10bS)-9-tert-butyl-5-phenyl-3,4,4a,5,6,10b...)
Affinity DataIC50:  300nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313420((4aS,5R,10bS)-9-tert-butyl-5-(5-chlorothiophen-2-y...)
Affinity DataIC50:  300nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313416((4aS,5R,10bS)-9-tert-butyl-5-(3-fluorophenyl)-3,4,...)
Affinity DataIC50:  350nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313388((4aS,5R,10bS)-5-phenyl-9-propyl-3,4,4a,5,6,10b-hex...)
Affinity DataIC50:  360nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313386((4aS,5R,10bS)-9-methyl-5-phenyl-3,4,4a,5,6,10b-hex...)
Affinity DataIC50:  420nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313395(2-((4aS,5R,10bS)-5-phenyl-3,4,4a,5,6,10b-hexahydro...)
Affinity DataIC50:  500nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313422((4aS,5R,10bS)-9-tert-butyl-5-(thiazol-2-yl)-3,4,4a...)
Affinity DataIC50:  530nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313402((4aS,5R,10bS)-8-chloro-7-fluoro-5-phenyl-3,4,4a,5,...)
Affinity DataIC50:  540nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313393((4aS,5R,10bS)-9-chloro-5-phenyl-3,4,4a,5,6,10b-hex...)
Affinity DataIC50:  720nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313416((4aS,5R,10bS)-9-tert-butyl-5-(3-fluorophenyl)-3,4,...)
Affinity DataIC50:  870nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313392((4aS,5R,10bS)-9-(pentafluoro-sulfanyl)-5-phenyl-2H...)
Affinity DataIC50:  910nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313423((4aS,5R,10bS)-9-tert-butyl-5-(pyridin-3-yl)-3,4,4a...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313403((4aS,5R,10bS)-8,9-dimethyl-5-phenyl-3,4,4a,5,6,10b...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313412(3-((4aS,5R,10bS)-9-tert-butyl-3,4,4a,5,6,10b-hexah...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313396((4aS,5R,10bS)-5-phenyl-9-(trifluoromethoxy)-3,4,4a...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50313398((4aS,5R,10bS)-N,N-dimethyl-5-phenyl-3,4,4a,5,6,10b...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of ATPase activity of human recombinant EG5 assessed as ATP hydrolysis by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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