Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]-4-DAMP from human muscarinic M3 receptor expressed in BHK-21 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-4-DAMP from human muscarinic M5 receptor expressed in BHK-21 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]-AFDX-384 from human muscarinic M2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-4-DAMP from human muscarinic M4 receptor expressed in BHK-21 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Agonist activity at human muscarinic M3 receptor expressed in BHK-21 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity to human adrenergic alpha1A receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to human adrenergic Alpha-1D receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Agonist activity at human muscarinic M5 receptor expressed in BHK-21 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Binding affinity to human adrenergic Alpha-1B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Displacement of [3H]-4-DAMP from human muscarinic M4 receptor expressed in BHK-21 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Binding affinity to human dopamine D2S receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Agonist activity at human muscarinic M5 receptor expressed in BHK-21 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Agonist activity at human muscarinic M3 receptor expressed in BHK-21 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Agonist activity at human muscarinic M2 receptor expressed in CHO-K1 cells coexpressing Galpha16 subunit assessed as increase of acetylcholine-induce...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Agonist activity at human muscarinic M4 receptor expressed in BHK-21 cells coexpressing Galpha16 subunit assessed as increase of acetylcholine-induce...More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Agonist activity at human muscarinic M2 receptor expressed in CHO-K1 cells coexpressing Galpha16 subunit assessed as increase of acetylcholine-induce...More data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Binding affinity to human adrenergic alpha1A receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Binding affinity to human 5-HT1A receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [3H]-4-DAMP from human muscarinic M4 receptor expressed in BHK-21 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Agonist activity at human muscarinic M2 receptor expressed in CHO-K1 cells coexpressing Galpha16 subunit assessed as increase of acetylcholine-induce...More data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Agonist activity at human muscarinic M3 receptor expressed in BHK-21 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Binding affinity to human adrenergic alpha2A receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 610nMAssay Description:Binding affinity to human histamine H1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 780nMAssay Description:Binding affinity to human histamine H1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Binding affinity to adrenergic alpha2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 910nMAssay Description:Binding affinity to human adrenergic Alpha-1B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 940nMAssay Description:Agonist activity at human muscarinic M5 receptor expressed in BHK-21 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 980nMAssay Description:Agonist activity at human muscarinic M2 receptor expressed in CHO-K1 cells coexpressing Galpha16 subunit assessed as increase of acetylcholine-induce...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
H. Lundbeck
Curated by ChEMBL
H. Lundbeck
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to ML2 (MT3) receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human choline transporter (CHT1) by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human neuropeptide Y1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human 5-HT transporter by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to I1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human NK1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human histamine H2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human MC4 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human 5-HT2A agonist site receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human 5-HT1A receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human muscarinic M1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human adenosine A1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human muscarinic M3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human adenosine A1 receptor agonist site by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human ETA receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human glucocorticoid receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human dopamine D3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human CCK2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to kappa opioid receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to adrenergic alpha2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to Lyn by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human dopamine D1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair