Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50039365
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335626((R)-2-((2-(3-Aminopiperidin-1-yl)-4-oxothieno[3,2-...)
Affinity DataIC50:  0.330nMAssay Description:Inhibition of DPP4 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335623((R)-2-((2-(3-Aminopiperidin-1-yl)-4-oxothieno-[2,3...)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of DPP4 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335624((R)-2-((2-(3-Aminopiperidin-1-yl)-5-methyl-4-oxoth...)
Affinity DataIC50:  1.32nMAssay Description:Inhibition of DPP4 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335627((R)-2-((2-(3-Aminopiperidin-1-yl)-7-methyl-4-oxoth...)
Affinity DataIC50:  1.72nMAssay Description:Inhibition of DPP4 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of DPP4 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335625((R)-2-((2-(3-Aminopiperidin-1-yl)-4-oxo-5-(trifluo...)
Affinity DataIC50:  88.8nMAssay Description:Inhibition of DPP4 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335623((R)-2-((2-(3-Aminopiperidin-1-yl)-4-oxothieno-[2,3...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP9 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335624((R)-2-((2-(3-Aminopiperidin-1-yl)-5-methyl-4-oxoth...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP9 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335625((R)-2-((2-(3-Aminopiperidin-1-yl)-4-oxo-5-(trifluo...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP9 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335626((R)-2-((2-(3-Aminopiperidin-1-yl)-4-oxothieno[3,2-...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP9 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335627((R)-2-((2-(3-Aminopiperidin-1-yl)-7-methyl-4-oxoth...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP9 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP8 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335627((R)-2-((2-(3-Aminopiperidin-1-yl)-7-methyl-4-oxoth...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP8 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335626((R)-2-((2-(3-Aminopiperidin-1-yl)-4-oxothieno[3,2-...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP8 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP9 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335624((R)-2-((2-(3-Aminopiperidin-1-yl)-5-methyl-4-oxoth...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP8 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335623((R)-2-((2-(3-Aminopiperidin-1-yl)-4-oxothieno-[2,3...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP8 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50335625((R)-2-((2-(3-Aminopiperidin-1-yl)-4-oxo-5-(trifluo...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of DPP8 after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed