Compile Data Set for Download or QSAR
maximum 50k data
Found 29 Enz. Inhib. hit(s) with all data for entry = 50032780
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataIC50:  366nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334557(CHEMBL1644513 | [4(5)S]-4(5)-(2-Aminoethyl)-2-(2-e...)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334550(CHEMBL1644506 | [4(5)R]-4(5)-(2-Aminoethyl)-2-[(3-...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334549(CHEMBL1644505 | [4(5)S]-4(5)-(2-Aminoethyl)-2-[(3-...)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334547(CHEMBL1644496 | [4(5)S]-4(5)-(2-Aminoethyl)-2-[(2,...)
Affinity DataIC50:  1.48E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334560(CHEMBL1644516 | [4(5)R]-4(5)-(2-Aminoethyl)-2-(2,3...)
Affinity DataIC50:  2.65E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334552(CHEMBL1644508 | [4(5)R]-4(5)-(2-Aminoethyl)-2-[(2,...)
Affinity DataIC50:  2.72E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334539((S)-4-(2-aminoethyl)-N-(2-bromophenyl)-4,5-dihydro...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334559(CHEMBL1644515 | [4(5)S]-4(5)-(2-Aminoethyl)-2-(2,3...)
Affinity DataIC50:  5.11E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334548(CHEMBL1644504 | [4(5)R]-4(5)-(2-Aminoethyl)-2-[(2,...)
Affinity DataIC50:  6.33E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334551(CHEMBL1644507 | [4(5)S]-4(5)-(2-Aminoethyl)-2-[(2,...)
Affinity DataIC50:  7.75E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334545(CHEMBL1644503 | [4(5)S]-4(5)-(2-Aminoethyl)-2-[(6-...)
Affinity DataIC50:  7.78E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334546(CHEMBL1644497 | [4(5)R]-4(5)-(2-Aminoethyl)-2-[(6-...)
Affinity DataIC50:  8.51E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334561(CHEMBL1644517 | [4(5)S]-4(5)-(2-Aminoethyl)-2-[(N-...)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334564(CHEMBL1644520 | [4(5)S]-4(5)-(2-Aminoethyl)-2-[(E)...)
Affinity DataIC50:  1.72E+4nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334558(CHEMBL1644514 | [4(5)R]-4(5)-(2-Aminoethyl)-2-(2-e...)
Affinity DataIC50:  3.25E+4nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334543((S)-4-(2-aminoethyl)-N-(3-chlorophenyl)-4,5-dihydr...)
Affinity DataIC50:  3.39E+4nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM85213(Agmatine | CAS_306-60-5 | CHEMBL58343 | NSC_199 | ...)
Affinity DataIC50:  3.65E+4nMAssay Description:Inhibition of Wistar rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334541((S)-4-(2-aminoethyl)-N-(4-bromophenyl)-4,5-dihydro...)
Affinity DataIC50:  5.94E+4nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334562(CHEMBL1644518 | [4(5)S]-4(5)-(2-Aminoethyl)-2-phen...)
Affinity DataIC50:  7.29E+4nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334542((S)-4-(2-aminoethyl)-N-(4-methoxyphenyl)-4,5-dihyd...)
Affinity DataIC50:  7.98E+4nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334540((S)-4-(2-aminoethyl)-N-(2,6-difluorophenyl)-4,5-di...)
Affinity DataIC50:  9.31E+4nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334553(CHEMBL1644509 | [4(5)S]-4(5)-(2-Aminoethyl)-2-[(di...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334555(CHEMBL1644511 | [4(5)S]-4(5)-(2-Aminoethyl)-2-[(na...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334538(CHEMBL1644495 | [4(5)S]-2-Benzylamino-4(5)-(2-amin...)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334563(CHEMBL1644519 | [4(5)S]-4(5)-(2-Aminoethyl)-2-(2-f...)
Affinity DataIC50:  1.17E+5nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334554(CHEMBL1644510 | [4(5)S]-4(5)-(2-Aminoethylo)-2-ben...)
Affinity DataIC50:  2.78E+5nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334556(CHEMBL1644512 | [4(5)R]-4(5)-(2-Aminoethyl)-2-[(na...)
Affinity DataIC50:  5.83E+5nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Gdansk University Of Technology

Curated by ChEMBL
LigandPNGBDBM50334544((S)-N-(4-(2-aminoethyl)-4,5-dihydro-1H-imidazol-2-...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed