TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 9.71E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at M5 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 6.54E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 5.22E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 3.79E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 3.21E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 2.19E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 5.37E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 1.85E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 5.10E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 4.40E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 3.07E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 1.38E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at M4 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology/Chemical Synthesis Core
Curated by ChEMBL
Affinity DataEC50: 5.82E+3nMAssay Description:Allosteric modulation at rat M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair