Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50033450
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50345577(CHEMBL1782082 | Hippolide A)
Affinity DataIC50:  2.38E+4nMAssay Description:Inhibition of recombinant PTP1B catalytic domain using pNPP as substrate assessed as pNP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50345576(CHEMBL1784622 | Hippolide B)
Affinity DataIC50:  3.97E+4nMAssay Description:Inhibition of recombinant PTP1B catalytic domain using pNPP as substrate assessed as pNP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50345578(CHEMBL1784623 | Hippolide E)
Affinity DataIC50:  4.04E+4nMAssay Description:Binding affinity at PKCalpha after 1 hr by luminescent kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50345577(CHEMBL1782082 | Hippolide A)
Affinity DataIC50:  6.20E+4nMAssay Description:Binding affinity at PKCgamma after 1 hr by luminescent kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed