TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Second Military Medical University
Curated by ChEMBL
Second Military Medical University
Curated by ChEMBL
Affinity DataIC50: 2.38E+4nMAssay Description:Inhibition of recombinant PTP1B catalytic domain using pNPP as substrate assessed as pNP releaseMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Second Military Medical University
Curated by ChEMBL
Second Military Medical University
Curated by ChEMBL
Affinity DataIC50: 3.97E+4nMAssay Description:Inhibition of recombinant PTP1B catalytic domain using pNPP as substrate assessed as pNP releaseMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Second Military Medical University
Curated by ChEMBL
Second Military Medical University
Curated by ChEMBL
Affinity DataIC50: 4.04E+4nMAssay Description:Binding affinity at PKCalpha after 1 hr by luminescent kinase assayMore data for this Ligand-Target Pair
TargetProtein kinase C gamma type(Homo sapiens (Human))
Second Military Medical University
Curated by ChEMBL
Second Military Medical University
Curated by ChEMBL
Affinity DataIC50: 6.20E+4nMAssay Description:Binding affinity at PKCgamma after 1 hr by luminescent kinase assayMore data for this Ligand-Target Pair