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Found 28 Enz. Inhib. hit(s) with all data for entry = 50033543
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347145(CHEMBL1797507)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347149(CHEMBL1797414)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347147(CHEMBL1797509)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347148(CHEMBL1797510)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337599((E/Z)-3-(3-(4-(3-phenylpropoxy)phenyl)allylamino)p...)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347149(CHEMBL1797414)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347150(CHEMBL1797499)
Affinity DataEC50:  6.70E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347151(CHEMBL1797500)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347152(CHEMBL1797501)
Affinity DataEC50:  7.20E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347153(CHEMBL1797502)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347154(CHEMBL1797503)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347155(CHEMBL1797504)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347156(CHEMBL1797505)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347157(CHEMBL1797506)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347145(CHEMBL1797507)
Affinity DataEC50:  7.80E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347146(CHEMBL1797508)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347147(CHEMBL1797509)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347148(CHEMBL1797510)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337599((E/Z)-3-(3-(4-(3-phenylpropoxy)phenyl)allylamino)p...)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347150(CHEMBL1797499)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347151(CHEMBL1797500)
Affinity DataEC50:  280nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347152(CHEMBL1797501)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347153(CHEMBL1797502)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347154(CHEMBL1797503)
Affinity DataEC50:  36nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347155(CHEMBL1797504)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347156(CHEMBL1797505)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347157(CHEMBL1797506)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50347146(CHEMBL1797508)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed