Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50034136
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research (Niper)

Curated by ChEMBL
LigandPNGBDBM50357677(CHEMBL1914951)
Affinity DataKi:  7.50E+4nMAssay Description:Competitive inhibition of human topoisomerase-2 alpha-ATPase activity by Lineweaver-Burk assay in presence of 200 to 520 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research (Niper)

Curated by ChEMBL
LigandPNGBDBM50357677(CHEMBL1914951)
Affinity DataIC50:  5.27E+4nMAssay Description:Inhibition of human topoisomerase 2 alpha-mediated decatenation of kDNA by agarose gel electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed