Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50033672
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349469(CHEMBL1808589)
Affinity DataIC50:  47nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349452(CHEMBL1808572)
Affinity DataIC50:  109nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349450(CHEMBL1808570)
Affinity DataIC50:  240nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349451(CHEMBL1808571)
Affinity DataIC50:  418nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349453(CHEMBL1808573)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349456(CHEMBL1808576)
Affinity DataIC50:  1.46E+3nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349454(CHEMBL1808574)
Affinity DataIC50:  1.73E+3nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349455(CHEMBL1808575)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349457(CHEMBL1808577)
Affinity DataIC50:  2.67E+3nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349467(CHEMBL1808587)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349449(CHEMBL1808569)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349468(CHEMBL1808588)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349458(CHEMBL1808578)
Affinity DataIC50:  4.94E+3nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349471(CHEMBL1808591)
Affinity DataIC50:  9.26E+3nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349461(CHEMBL1808581)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349470(CHEMBL1808590)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349466(CHEMBL1808586)
Affinity DataIC50:  1.87E+4nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349459(CHEMBL1808579)
Affinity DataIC50:  2.07E+4nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349460(CHEMBL1808580)
Affinity DataIC50:  2.14E+4nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349462(CHEMBL1808582)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349465(CHEMBL1808585)
Affinity DataIC50:  2.83E+4nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349464(CHEMBL1808584)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349463(CHEMBL1808583)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349476(CHEMBL1808596)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349472(CHEMBL1808592)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349473(CHEMBL1808593)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349474(CHEMBL1808594)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50349475(CHEMBL1808595)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed