Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50033818
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universita` Degli Studi Di Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50048866(1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydro-na...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor from guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universita` Degli Studi Di Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50035131((+)-(6R,11S)-6,11-dimethyl-3-(3-methyl-but-2-enyl)...)
Affinity DataKi:  2.62nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor from guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universita` Degli Studi Di Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50351992(CHEMBL1822599)
Affinity DataKi:  9.08nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor from guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universita` Degli Studi Di Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50351993(CHEMBL1822600)
Affinity DataKi:  19.8nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor from guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universita` Degli Studi Di Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50351990(CHEMBL1822597)
Affinity DataKi:  78.7nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor from guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universita` Degli Studi Di Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50351991(CHEMBL1822598)
Affinity DataKi:  96.2nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor from guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universita` Degli Studi Di Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50351988(CHEMBL1822595)
Affinity DataKi:  2.57E+3nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor from guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universita` Degli Studi Di Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50351989(CHEMBL1822596)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor from guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed