Compile Data Set for Download or QSAR
maximum 50k data
Found 51 Enz. Inhib. hit(s) with all data for entry = 50034047
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]testosterone from androgen receptor in Sprague-Dawley rat prostate gland after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataIC50:  3.10nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50338693(2-methyl-2-((3aR,4S,9bS)-8-nitro-3a,4,5,9b-tetrahy...)
Affinity DataIC50:  5.10nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Oryctolagus cuniculus)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM8903((1S,2R,10S,11S,14S,15S)-14-acetyl-2,15-dimethyltet...)
Affinity DataIC50:  6nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355949(CHEMBL1910418)
Affinity DataIC50:  22nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataIC50:  22nMAssay Description:Displacement of [3H]Dex from glucocorticoid receptor in Sprague-Dawley rat liver after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]testosterone from androgen receptor in Sprague-Dawley rat prostate gland after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50:  26nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355938(CHEMBL1909642)
Affinity DataIC50:  38nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(RAT)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM19214((1S,2R,10S,11S,14S,15R,17S)-17-hydroxy-14-(2-hydro...)
Affinity DataIC50:  43nMAssay Description:Displacement of [3H]Aldo from mineralocorticoid receptor in Sprague-Dawley rat kidney after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50:  45nMAssay Description:Displacement of [3H]testosterone from androgen receptor in Sprague-Dawley rat prostate gland after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355940(CHEMBL1910408)
Affinity DataIC50:  45nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355937(CHEMBL1910406)
Affinity DataIC50:  59nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355950(CHEMBL1910419)
Affinity DataIC50:  89nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355942(CHEMBL1910410)
Affinity DataIC50:  100nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Oryctolagus cuniculus)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataIC50:  440nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355941(CHEMBL1910409)
Affinity DataIC50: >1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355939(CHEMBL1910407)
Affinity DataIC50: >1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355951(CHEMBL1910420)
Affinity DataIC50: >1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355948(CHEMBL1910417)
Affinity DataIC50: >1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355947(CHEMBL1910416)
Affinity DataIC50: >1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355943(CHEMBL1910412)
Affinity DataIC50: >1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355944(CHEMBL1910413)
Affinity DataIC50: >1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355945(CHEMBL1910414)
Affinity DataIC50: >1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355946(CHEMBL1910415)
Affinity DataIC50: >1.00E+3nMAssay Description:Competitive binding affinity to rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355938(CHEMBL1909642)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(RAT)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataIC50:  2.10E+3nMAssay Description:Displacement of [3H]Aldo from mineralocorticoid receptor in Sprague-Dawley rat kidney after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Oryctolagus cuniculus)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50:  3.40E+3nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Oryctolagus cuniculus)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)
Affinity DataIC50:  5.60E+3nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355950(CHEMBL1910419)
Affinity DataIC50:  8.00E+3nMAssay Description:Antagonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355942(CHEMBL1910410)
Affinity DataIC50:  1.40E+4nMAssay Description:Antagonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(RAT)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50:  1.40E+4nMAssay Description:Displacement of [3H]Aldo from mineralocorticoid receptor in Sprague-Dawley rat kidney after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataIC50:  2.00E+4nMAssay Description:Displacement of [3H]Dex from glucocorticoid receptor in Sprague-Dawley rat liver after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355949(CHEMBL1910418)
Affinity DataIC50:  2.90E+4nMAssay Description:Antagonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355940(CHEMBL1910408)
Affinity DataIC50:  4.40E+4nMAssay Description:Antagonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50:  4.90E+4nMAssay Description:Displacement of [3H]Dex from glucocorticoid receptor in Sprague-Dawley rat liver after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355937(CHEMBL1910406)
Affinity DataIC50:  6.10E+4nMAssay Description:Antagonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]E2 from estrogen receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)
Affinity DataIC50:  3.20E+5nMAssay Description:Displacement of [3H]Dex from glucocorticoid receptor in Sprague-Dawley rat liver after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(RAT)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataIC50:  3.40E+5nMAssay Description:Displacement of [3H]E2 from estrogen receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(RAT)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)
Affinity DataIC50:  3.60E+5nMAssay Description:Displacement of [3H]Aldo from mineralocorticoid receptor in Sprague-Dawley rat kidney after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(RAT)
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)
Affinity DataIC50: >1.00E+6nMAssay Description:Displacement of [3H]E2 from estrogen receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataEC50:  0.970nMAssay Description:Agonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50338693(2-methyl-2-((3aR,4S,9bS)-8-nitro-3a,4,5,9b-tetrahy...)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355937(CHEMBL1910406)
Affinity DataEC50:  95nMAssay Description:Agonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355950(CHEMBL1910419)
Affinity DataEC50:  46nMAssay Description:Agonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355949(CHEMBL1910418)
Affinity DataEC50:  75nMAssay Description:Agonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355936(CHEMBL1910411)
Affinity DataEC50:  13nMAssay Description:Agonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355938(CHEMBL1909642)
Affinity DataEC50:  190nMAssay Description:Agonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50355940(CHEMBL1910408)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at rat androgen receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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