Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50042308
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423866(CHEMBL2024148)
Affinity DataKd:  17nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423867(CHEMBL2023737)
Affinity DataKd:  21nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423868(CHEMBL2023738)
Affinity DataKd:  0.331nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423869(CHEMBL2023739)
Affinity DataKd:  1.5nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423870(CHEMBL2024147)
Affinity DataKd:  38nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423872(CHEMBL2024150)
Affinity DataKd:  166nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO cells assessed as inhibition of NECA-induced increase of intracellular cAMP level...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423872(CHEMBL2024150)
Affinity DataKd:  3.40nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423873(CHEMBL2024151)
Affinity DataKd:  148nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423874(CHEMBL2024152)
Affinity DataKd:  5.60nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423871(CHEMBL2024149)
Affinity DataKd:  275nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO cells assessed as inhibition of NECA-induced increase of intracellular cAMP level...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423871(CHEMBL2024149)
Affinity DataKd:  0.437nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NECA-induced CRE-SPAP gene t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed